SCHEMBL4848831

SCHEMBL4848831

O=C(O)c1cc(F)cc(N2CCCOCC2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.55
TTR P02766 1/20 0.49
ALDH1A1 P00352 3/20 0.44
HPGD P15428 3/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GPR183 P32249 1/20 0.44
DDR2 Q16832 1/20 0.44
POLB P06746 1/20 0.43
PIK3CA P42336 2/20 0.43
AKR1C3 P42330 2/20 0.41
MAPT P10636 4/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
NPSR1 Q6W5P4 2/20 0.41
BRAF P15056 2/20 0.41
TP53 P04637 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593762 0.94 KMO (0.60) KMOTTRALDH1A1HPGDGPR183
SCHEMBL594366 0.86 ALDH1A1 (0.57) KMOTTRALDH1A1HPGDKDM4E
SCHEMBL594127 0.85 KDM4E (0.56) KMOTTRALDH1A1HPGDKDM4E
SCHEMBL592613 0.85 KDM4E (0.56) KMOTTRALDH1A1HPGDKDM4E
SCHEMBL27893364 0.83 KMO (0.70) KMOALDH1A1HPGDKDM4EMEN1
SCHEMBL6629680 0.81 MAPT (0.49) KMOTTRALDH1A1KDM4EGPR183
SCHEMBL1793059 0.81 KMO (0.48) KMOALDH1A1HPGDMEN1KMT2A
SCHEMBL4757032 0.77 KMO (0.62) KMOALDH1A1HPGDMEN1KMT2A
SCHEMBL23662606 0.77 MRGPRX4 (0.49) KMOALDH1A1HPGDKDM4EMEN1
SCHEMBL593990 0.76 TTR (0.53) KMOTTRALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed
WO-2007075896-A2 HETEROCYCLIC CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-07-05 WO disclosed