SCHEMBL4853541

SCHEMBL4853541

Cc1ccc(OCCN(C)C)c(C(=O)/C=C/c2ccc(O)c(F)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.53
SNCA P37840 1/20 0.44
MAOB P27338 1/20 0.44
MAPT P10636 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4854223 1.00 MCL1 (0.53) MCL1SNCAMAOBMAPTMAPK1
SCHEMBL4847824 0.90 TUBB1 (0.55) MCL1MAPTKMT2ABCHEACHE
SCHEMBL4853445 0.90 TUBB1 (0.55) MCL1MAPTKMT2ABCHEACHE
SCHEMBL4851370 0.89 MCL1 (0.48) MCL1MAOBKMT2ABCHEACHE
SCHEMBL4847316 0.89 MCL1 (0.48) MCL1MAOBKMT2ABCHEACHE
SCHEMBL4856299 0.87 MCL1 (0.50) MCL1SNCAMAOBKMT2ABCHE
SCHEMBL4854973 0.87 MCL1 (0.50) MCL1SNCAMAOBKMT2ABCHE
SCHEMBL4850004 0.83 TUBB4A (0.55) MCL1MAOBMAPTKMT2ABCHE
SCHEMBL4854901 0.83 TUBB4A (0.55) MCL1MAOBMAPTKMT2ABCHE
SCHEMBL4853546 0.80 SNCA (0.48) SNCABCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed