SCHEMBL4856299

SCHEMBL4856299

CN(C)CCOc1ccc(C(C)(C)C)cc1C(=O)C=Cc1ccc(O)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.50
KDM4E B2RXH2 1/20 0.46
ESR1 P03372 2/20 0.42
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
TUBB1 Q9H4B7 1/20 0.41
CXCL12 P48061 2/20 0.40
TNFRSF1A P19438 1/20 0.40
MAOB P27338 1/20 0.40
SNCA P37840 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4854973 1.00 MCL1 (0.50) MCL1KDM4EESR1BCHEACHE
SCHEMBL4852536 0.90 TUBB1 (0.53) MCL1KDM4EBCHEACHEMEN1
SCHEMBL4853707 0.90 TUBB1 (0.53) MCL1KDM4EBCHEACHEMEN1
SCHEMBL4853541 0.87 MCL1 (0.53) MCL1BCHEACHEKMT2AMAOB
SCHEMBL4854223 0.87 MCL1 (0.53) MCL1BCHEACHEKMT2AMAOB
SCHEMBL4849818 0.87 KDM4E (0.51) MCL1KDM4EBCHEACHELMNA
SCHEMBL4849756 0.87 KDM4E (0.51) MCL1KDM4EBCHEACHELMNA
SCHEMBL4847316 0.83 MCL1 (0.48) MCL1BCHEACHEMEN1LMNA
SCHEMBL4851370 0.83 MCL1 (0.48) MCL1BCHEACHEMEN1LMNA
SCHEMBL4854982 0.82 KDM4E (0.47) KDM4EESR1BCHEACHESNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed