SCHEMBL4853553

SCHEMBL4853553

CCOC(=O)COc1c(C)cc(NC(=O)OC(C)(C)C)cc1C

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 8/20 0.45
ALDH1A1 P00352 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA9 Q16790 1/20 0.41
PPARG P37231 1/20 0.41
KDM4E B2RXH2 1/20 0.40
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
IDH1 O75874 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTT P42858 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ESR1 P03372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7387537 0.87 NLRP3 (0.54) NLRP3ALDH1A1KDM4ECYP1A2CYP2C19
SCHEMBL4855183 0.83 ESR1 (0.51) NLRP3ALDH1A1CA12CA1CA9
SCHEMBL2847349 0.82 AAK1 (0.43) NLRP3ALDH1A1CA12CA1CA9
SCHEMBL8649013 0.82 NLRP3 (0.46) NLRP3ALDH1A1KDM4EMEN1KMT2A
SCHEMBL1549923 0.80 NLRP3 (0.48) NLRP3ALDH1A1KDM4ECYP1A2CYP2C19
SCHEMBL4856473 0.80 EPHX2 (0.54) ALDH1A1PPARGKDM4ECYP1A2IDH1
SCHEMBL7390785 0.79 NLRP3 (0.46) NLRP3ALDH1A1KDM4ECYP1A2CYP2C19
SCHEMBL8194998 0.78 CD69 (0.46) NLRP3ALDH1A1CA12CA9KDM4E
SCHEMBL7475639 0.78 SMN1; SMN2 (0.56) ALDH1A1PPARGCYP1A2CYP2C19IDH1
SCHEMBL16302366 0.77 CA12 (0.51) ALDH1A1CA12CA1CA9KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7345067-B2 Aniline derivatives, their manufacture and use as pharmaceutical agents HOFFMANN-LA ROCHE INC. (US) 2008-03-18 US disclosed
US-20040248951-A1 Aniline derivatives, their manufacture and use as pharmaceuticals F. HOFFMANN-LA ROCHE AG, A SWISS COMPANY (CH) 2004-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040248951-A1 Aniline derivatives, their manufacture and use as pharmaceuticals PPARA, PPARD, PPARG NLRP3 4061/4885ALDH1A1 464/4885CA12 4686/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.