SCHEMBL1549923

SCHEMBL1549923

CCOC(=O)COc1c(C)cc(NC)cc1C

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 7/20 0.48
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43
GAA P10253 3/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7387537 0.89 NLRP3 (0.54) NLRP3ALDH1A1CYP1A2CYP2C19KDM4E
SCHEMBL7394140 0.83 NLRP3 (0.57) NLRP3ALDH1A1CYP1A2CYP2C19GAA
SCHEMBL29485565 0.83 ALDH1A1 (0.47) NLRP3ALDH1A1CYP1A2CYP2C19GAA
SCHEMBL7390785 0.81 NLRP3 (0.46) NLRP3ALDH1A1CYP1A2CYP2C19GAA
SCHEMBL1549815 0.80 ESR1 (0.54) ALDH1A1CYP1A2NPSR1KDM4EHSD17B10
SCHEMBL7386523 0.80 ATM (0.47) NLRP3ALDH1A1CYP1A2CYP2C19GAA
SCHEMBL7028752 0.80 ALDH1A1 (0.58) NLRP3ALDH1A1CYP1A2CYP2C19GAA
SCHEMBL4853186 0.80 ALDH1A1 (0.45) NLRP3ALDH1A1CYP1A2CYP2C19GAA
SCHEMBL4853553 0.80 NLRP3 (0.45) NLRP3ALDH1A1CYP1A2CYP2C19KDM4E
SCHEMBL8194998 0.79 CD69 (0.46) NLRP3ALDH1A1CYP1A2CYP2C19GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2314576-A1 Phenyl derivatives as PPAR agonists F.HOFFMANN-LA ROCHE AG (CH) 2011-04-27 EP disclosed
US-7112599-B2 Oxazole compounds for the treatment of neurodegenerative disorders PFIZER INC. (US) 2006-09-26 US disclosed
EP-1682508-A1 PHENYL DERIVATIVES AS PPAR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049573-A1 PHENYL DERIVATIVES AS PPAR AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed
US-5905068-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1999-05-18 US disclosed