SCHEMBL4853728

SCHEMBL4853728

C=CC(=O)n1c[c]c2ccccc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
AKT1 P31749 1/20 0.33
KRAS P01116 1/20 0.33
ACHE P22303 4/20 0.33
KMT2A Q03164 2/20 0.33
TET3 O43151 1/20 0.33
FBXL19 Q6PCT2 1/20 0.33
CXXC5 Q7LFL8 1/20 0.33
TET1 Q8NFU7 1/20 0.33
KDM2B Q8NHM5 1/20 0.33
CXXC4 Q9H2H0 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
TGM2 P21980 1/20 0.31
GSK3B P49841 1/20 0.31
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
HTT P42858 1/20 0.30
PAX8 Q06710 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8871120 0.78 TSHR (0.34) TSHRKMT2AALDH1A1
SCHEMBL9581907 0.72 KMT2A (0.46) CYP2D6TSHRKMT2AMEN1ALDH1A1
SCHEMBL9582187 0.70 ALDH1A1 (0.43) TSHRKMT2AMEN1ALDH1A1GAA
SCHEMBL1948855 0.69 BCHE (0.44) KMT2AMEN1ALDH1A1
SCHEMBL10835083 0.68 NOTUM (0.59) TSHRKMT2AMEN1ALDH1A1GAA
SCHEMBL31565005 0.68 NOTUM (0.59) TSHRKMT2AMEN1ALDH1A1GAA
SCHEMBL29182109 0.66 KMT2A (0.53) KMT2AMEN1ALDH1A1HTT
SCHEMBL5373174 0.65 KDM4E (0.34)
SCHEMBL32689427 0.64 POLB (0.55) KRASKMT2AMEN1ALDH1A1GAA
SCHEMBL811819 0.64 POLB (0.55) KRASKMT2AMEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008144263-A1 POTENT INDOLE-3-CARBINOL-DERIVED ANTITUMOR AGENTS THE OHIO STATE UNIVERSITY RESEARCH FOUNDATION (US) 2008-11-27 WO disclosed