SCHEMBL10835083

SCHEMBL10835083

C=CC(=O)n1ccc2ccccc21

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.59
TSHR P16473 2/20 0.56
RAB9A P51151 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
KMT2A Q03164 3/20 0.43
TFPI2 P48307 1/20 0.42
NPY4R P50391 1/20 0.42
GAA P10253 1/20 0.42
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
LMNA P02545 2/20 0.40
CDK4 P11802 3/20 0.38
CCND1 P24385 3/20 0.38
MAPK1 P28482 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31565005 1.00 NOTUM (0.59) NOTUMTSHRRAB9AL3MBTL1KMT2A
SCHEMBL1527302 0.79 NOTUM (0.52) NOTUMTSHRRAB9AL3MBTL1KMT2A
SCHEMBL3397331 0.79 NOTUM (0.56) NOTUMTSHRRAB9AL3MBTL1KMT2A
SCHEMBL14272674 0.78 NOTUM (0.51) NOTUMTSHRRAB9AL3MBTL1KMT2A
SCHEMBL1151123 0.78 NOTUM (0.70) NOTUMTSHRRAB9AL3MBTL1KMT2A
SCHEMBL10477477 0.78 NOTUM (0.70) NOTUMTSHRRAB9AL3MBTL1KMT2A
SCHEMBL29453277 0.76 TSHR (0.69) NOTUMTSHRRAB9AL3MBTL1KMT2A
SCHEMBL931955 0.76 TSHR (0.69) NOTUMTSHRRAB9AL3MBTL1KMT2A
SCHEMBL21808239 0.76 KRAS (0.50)
SCHEMBL20905232 0.76 TFPI2 (0.47) NOTUMTFPI2ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1709921-A Resin of zinc acrylate or copper acrylate containing indole function group, its preparation and use CHINESE OCEANOGRAPHY UNIV (CN) 2005-12-21 CN claimed
US-20250120982-A1 COVALENT TARGETING OF E3 LIGASES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2025-04-17 US disclosed
US-12161648-B2 Covalent targeting of E3 ligases THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-12-10 US disclosed
WO-2024097262-A1 CHEMOPROTEOMIC CAPTURE OF RNA BINDING ACTIVITY IN LIVING CELLS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2024-05-10 WO disclosed
US-20240103005-A1 N-ACRYLOYLINDOLES AND METHODS OF USE VERSITECH LIMITED (CN) 2024-03-28 US disclosed
US-20240103005-A1 N-ACRYLOYLINDOLES AND METHODS OF USE VERSITECH LIMITED (CN) 2024-03-28 US disclosed
CN-117126096-A N-acryloylindoles and methods of use 香港大学 2023-11-28 CN disclosed
CN-117126096-A N-acryloylindoles and methods of use 香港大学 2023-11-28 CN disclosed
CN-117126096-A N-acryloylindoles and methods of use 香港大学 2023-11-28 CN disclosed
US-11666661-B2 Methods and compounds for targeted autophagy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-06-06 US disclosed
US-20190290778-A1 METHODS AND COMPOUNDS FOR TARGETED AUTOPHAGY FRONTIER MEDICINES CORPORATION 2019-09-26 US disclosed
WO-2019183600-A1 METHODS AND COMPOUNDS FOR TARGETED AUTOPHAGY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-09-26 WO disclosed
WO-2019075386-A1 MTORC1 MODULATORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-04-18 WO disclosed
US-20190112268-A1 mTORC1 MODULATORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2019-04-18 US disclosed
CN-1709921-B Resin of zinc acrylate or copper acrylate containing indole function group, its preparation and use OCEAN UNIV CHINA 2011-09-28 CN disclosed
CN-1709921-A Resin of zinc acrylate or copper acrylate containing indole function group, its preparation and use CHINESE OCEANOGRAPHY UNIV (CN) 2005-12-21 CN disclosed
EP-0091039-B1 ANTI-FOULING AGENT Nitto Kasei Co., Ltd. (JP) 1986-10-01 EP disclosed
US-4598156-A Process for producing indoles unsubstituted in the 2,3-position and N(3-chloropropionyl)indole produced thereby CIBA GEIGY CORPORATION (US) 1986-07-01 US disclosed
US-4526932-A Copolymer containing N-coordinated triorganotin compound NITTO KASEI CO., LTD. (JP) 1985-07-02 US disclosed
EP-0091039-A2 Anti-fouling agent Nitto Kasei Co., Ltd. (JP) 1983-10-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240103005-A1 N-ACRYLOYLINDOLES AND METHODS OF USE NAT1, DDIT3, ACR NOTUM 3260/4885TSHR 3784/4885RAB9A 3380/4885
US-12161648-B2 Covalent targeting of E3 ligases RNF114, RNF4, RNF168 NOTUM 2977/4885TSHR 4065/4885RAB9A 2224/4885
US-20190290778-A1 METHODS AND COMPOUNDS FOR TARGETED AUTOPHAGY ATG7, BECN1, SQSTM1 NOTUM 4238/4885TSHR 4601/4885RAB9A 223/4885
US-20190112268-A1 mTORC1 MODULATORS MTOR, RPTOR, RICTOR NOTUM 3808/4885TSHR 3686/4885RAB9A 439/4885
US-11666661-B2 Methods and compounds for targeted autophagy ATG7, BECN1, SQSTM1 NOTUM 4238/4885TSHR 4601/4885RAB9A 223/4885
US-20250120982-A1 COVALENT TARGETING OF E3 LIGASES STUB1, XIAP, RBX1 NOTUM 3544/4885TSHR 4386/4885RAB9A 2030/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.