SCHEMBL4853801

SCHEMBL4853801

CN(C)CCNc1ccc(C(=O)C=Cc2cc(-c3ccccc3)ccc2OCCN(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 9/20 0.53
BCHE P06276 6/20 0.50
ACHE P22303 6/20 0.50
TNFRSF1A P19438 1/20 0.44
KDR P35968 1/20 0.44
SLC6A9 P48067 1/20 0.43
HTR2C P28335 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3684939 0.91 TNFRSF1A (0.54) MCHR1BCHETNFRSF1A
SCHEMBL4847749 0.90 ACHE (0.42) MCHR1BCHEACHETNFRSF1AKDR
SCHEMBL4848121 0.87 BCHE (0.55) MCHR1BCHEACHETNFRSF1ASLC6A9
SCHEMBL4849165 0.85 BCHE (0.58) MCHR1BCHEACHETNFRSF1A
SCHEMBL4856388 0.84 BCHE (0.49) MCHR1BCHEACHESLC6A9
SCHEMBL4853797 0.84 BCHE (0.49) MCHR1BCHEACHESLC6A9
SCHEMBL4852888 0.81 HCRTR2 (0.42) MCHR1BCHEACHETNFRSF1AKDR
SCHEMBL4853736 0.81 BCHE (0.52) MCHR1BCHEACHETNFRSF1ASLC6A9
SCHEMBL14280889 0.80 BCHE (0.53) MCHR1BCHEACHETNFRSF1ASLC6A9
SCHEMBL4853884 0.80 BCHE (0.53) MCHR1BCHEACHETNFRSF1ASLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed