SCHEMBL4848121

SCHEMBL4848121

CN(C)CCOc1ccc(-c2ccccc2)cc1C=CC(=O)c1ccc(O)cc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BCHE P06276 5/20 0.55
ACHE P22303 5/20 0.55
CAPN1 P07384 2/20 0.51
MCHR1 Q99705 1/20 0.50
MAOB P27338 1/20 0.48
CTSL P07711 2/20 0.47
CTSB P07858 2/20 0.47
SLC6A9 P48067 2/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TNFRSF1A P19438 1/20 0.45
DPP4 P27487 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4849165 0.90 BCHE (0.58) BCHEACHEMCHR1MAOBALDH1A1
SCHEMBL4852218 0.88 CAPN1 (0.50) BCHEACHECAPN1MAOBCTSL
SCHEMBL4853801 0.87 MCHR1 (0.53) BCHEACHEMCHR1SLC6A9TNFRSF1A
SCHEMBL4853736 0.85 BCHE (0.52) BCHEACHEMCHR1SLC6A9KDM4E
SCHEMBL14280889 0.84 BCHE (0.53) BCHEACHEMCHR1SLC6A9KDM4E
SCHEMBL4853884 0.84 BCHE (0.53) BCHEACHEMCHR1SLC6A9KDM4E
SCHEMBL4848110 0.82 BCHE (0.51) BCHEACHECAPN1MCHR1MAOB
SCHEMBL4853434 0.82 BCHE (0.51) BCHEACHECAPN1MCHR1MAOB
SCHEMBL4849762 0.82 KDM4E (0.52) BCHEACHECAPN1MAOBCTSL
SCHEMBL14280884 0.80 BCHE (0.46) BCHEACHECAPN1CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed