SCHEMBL4854470

SCHEMBL4854470

Cc1ccccc1-c1ccc(OCCCCN(C)C)c(C=CC(=O)c2ccccc2CN(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
HRH1 P35367 2/20 0.40
SLC6A9 P48067 2/20 0.40
BCHE P06276 8/20 0.40
ACHE P22303 7/20 0.40
PTPN11 Q06124 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NMT2 O60551 1/20 0.37
NMT1 P30419 1/20 0.37
PTPN1 P18031 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4847450 0.94 SLC6A9 (0.43) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4845311 0.93 MAOB (0.42) BCHEACHE
SCHEMBL4852923 0.92 SLC6A9 (0.37) KDM4ESLC6A9BCHEACHEPTPN11
SCHEMBL4853384 0.92 PTPN11 (0.37) KDM4ESLC6A9BCHEACHEPTPN11
SCHEMBL4848040 0.90 HRH1 (0.39) KDM4EHRH1SLC6A9PTPN11NMT2
SCHEMBL4854469 0.90 SLC6A9 (0.43) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4856457 0.90 SLC6A9 (0.43) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4849688 0.89 SLC6A9 (0.41) KDM4ESLC6A9BCHEACHEALDH1A1
SCHEMBL4852335 0.89 SLC6A9 (0.40) KDM4EHRH1SLC6A9BCHEACHE
SCHEMBL4854695 0.88 SLC6A9 (0.43) KDM4EHRH1SLC6A9BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed