SCHEMBL4852335

SCHEMBL4852335

Cc1ccccc1-c1ccc(OCCN(C)C(C)(C)C)c(C=CC(=O)c2ccccc2CN(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 5/20 0.40
MCHR1 Q99705 1/20 0.37
NMT2 O60551 1/20 0.36
NMT1 P30419 1/20 0.36
PTPN1 P18031 2/20 0.35
HRH1 P35367 1/20 0.35
TNFRSF1A P19438 2/20 0.35
MAOB P27338 1/20 0.35
TUBB4A P04350 2/20 0.34
TUBB P07437 2/20 0.34
TUBA3C P0DPH7 2/20 0.34
TUBA1B P68363 2/20 0.34
TUBA4A P68366 2/20 0.34
TUBB4B P68371 2/20 0.34
TUBB3 Q13509 2/20 0.34
TUBB2A Q13885 2/20 0.34
TUBB8 Q3ZCM7 2/20 0.34
TUBA3E Q6PEY2 2/20 0.34
TUBA1A Q71U36 2/20 0.34
TUBA1C Q9BQE3 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852923 0.95 SLC6A9 (0.37) SLC6A9MCHR1NMT2NMT1PTPN1
SCHEMBL4853384 0.94 PTPN11 (0.37) SLC6A9NMT2NMT1PTPN1TNFRSF1A
SCHEMBL4853580 0.93 SLC6A9 (0.40) SLC6A9MCHR1PTPN1HRH1TNFRSF1A
SCHEMBL4847450 0.92 SLC6A9 (0.43) SLC6A9MCHR1NMT2NMT1PTPN1
SCHEMBL4852352 0.91 SLC6A9 (0.43) SLC6A9MCHR1NMT2NMT1PTPN1
SCHEMBL4847208 0.91 SLC6A9 (0.43) SLC6A9MCHR1NMT2NMT1PTPN1
SCHEMBL4849688 0.89 SLC6A9 (0.41) SLC6A9MCHR1MAOBKDM4EALDH1A1
SCHEMBL4854470 0.89 KDM4E (0.43) SLC6A9NMT2NMT1PTPN1HRH1
SCHEMBL4854695 0.86 SLC6A9 (0.43) SLC6A9MCHR1NMT2NMT1HRH1
SCHEMBL4852369 0.86 HRH1 (0.41) SLC6A9MCHR1NMT2NMT1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed