SCHEMBL4853384

SCHEMBL4853384

Cc1ccccc1-c1ccc(OCCCCCN(C)C(C)(C)C)c(C=CC(=O)c2ccccc2CN(C)C)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.37
SLC6A9 P48067 2/20 0.37
MAOB P27338 4/20 0.36
MAOA P21397 3/20 0.36
APP P05067 2/20 0.36
PTPN1 P18031 1/20 0.36
BCHE P06276 7/20 0.35
ACHE P22303 6/20 0.35
TNFRSF1A P19438 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NMT2 O60551 1/20 0.34
NMT1 P30419 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852923 0.99 SLC6A9 (0.37) PTPN11SLC6A9MAOBMAOAAPP
SCHEMBL4852335 0.94 SLC6A9 (0.40) SLC6A9MAOBPTPN1BCHEACHE
SCHEMBL4854470 0.92 KDM4E (0.43) PTPN11SLC6A9PTPN1BCHEACHE
SCHEMBL4853380 0.91 SLC6A9 (0.40) PTPN11SLC6A9MAOBMAOAAPP
SCHEMBL4854641 0.91 SLC6A9 (0.40) PTPN11SLC6A9MAOBMAOAAPP
SCHEMBL4853354 0.90 SLC6A9 (0.40) PTPN11SLC6A9MAOBMAOAAPP
SCHEMBL4852918 0.90 SLC6A9 (0.40) PTPN11SLC6A9MAOBMAOAAPP
SCHEMBL4853580 0.89 SLC6A9 (0.40) SLC6A9MAOBPTPN1BCHEACHE
SCHEMBL4845311 0.88 MAOB (0.42) MAOBMAOAAPPBCHEACHE
SCHEMBL4847450 0.88 SLC6A9 (0.43) SLC6A9PTPN1BCHEACHEKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed