SCHEMBL4854964

SCHEMBL4854964

Cc1ccccc1-c1ccc(OCCN(C)C)c(C=CC(=O)c2cccc(CN(C)C)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.43
SLC6A9 P48067 2/20 0.42
HTR7 P34969 2/20 0.41
HRH1 P35367 1/20 0.41
ACHE P22303 1/20 0.41
TNFRSF1A P19438 6/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PTPN1 P18031 1/20 0.39
MCHR1 Q99705 1/20 0.38
ESR1 P03372 1/20 0.37
FFAR1 O14842 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4851258 0.91 BCHE (0.47) BCHESLC6A9HRH1ACHETNFRSF1A
SCHEMBL14280889 0.89 BCHE (0.53) BCHESLC6A9HRH1ACHETNFRSF1A
SCHEMBL4853884 0.89 BCHE (0.53) BCHESLC6A9HRH1ACHETNFRSF1A
SCHEMBL4846169 0.87 BCHE (0.42) BCHEHRH1ACHETNFRSF1AKDM4E
SCHEMBL4848150 0.86 BCHE (0.42) BCHESLC6A9HRH1ACHETNFRSF1A
SCHEMBL4852794 0.86 MCHR1 (0.45) BCHESLC6A9ACHETNFRSF1AALDH1A1
SCHEMBL4847357 0.84 NR1H4 (0.50) BCHEHRH1ACHEKDM4EALDH1A1
SCHEMBL4854809 0.84 NR1H4 (0.50) BCHEHRH1ACHEKDM4EALDH1A1
SCHEMBL4856336 0.84 LMNA (0.46) BCHESLC6A9ACHEKDM4EALDH1A1
SCHEMBL4856323 0.84 LMNA (0.46) BCHESLC6A9ACHEKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed