SCHEMBL4846169

SCHEMBL4846169

Cc1cc(C)cc(-c2ccc(OCCN(C)C)c(C=CC(=O)c3cccc(CN(C)C)c3)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.42
ACHE P22303 1/20 0.40
TNFRSF1A P19438 10/20 0.39
PTPN1 P18031 1/20 0.38
HRH1 P35367 1/20 0.38
KDR P35968 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4853884 0.90 BCHE (0.53) BCHEACHETNFRSF1APTPN1HRH1
SCHEMBL14280889 0.90 BCHE (0.53) BCHEACHETNFRSF1APTPN1HRH1
SCHEMBL4853514 0.89 NR1H4 (0.47) BCHEACHEKDR
SCHEMBL4853736 0.88 BCHE (0.52) BCHEACHETNFRSF1AHRH1KDM4E
SCHEMBL4856637 0.88 LMNA (0.45) BCHEACHETNFRSF1APTPN1KDR
SCHEMBL4853345 0.88 RELA (0.48) BCHEACHETNFRSF1APTPN1KDR
SCHEMBL4854964 0.87 BCHE (0.43) BCHEACHETNFRSF1APTPN1HRH1
SCHEMBL4847119 0.85 SNCA (0.41) BCHEACHETNFRSF1APTPN1
SCHEMBL4847433 0.85 TNFRSF1A (0.46) TNFRSF1APTPN1
SCHEMBL4846042 0.84 MAPT (0.50) BCHEACHEKDRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed