SCHEMBL4854982

SCHEMBL4854982

CN(C)CCOc1ccc(C(C)(C)C)cc1C=CC(=O)c1ccc(O)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.47
SNCA P37840 2/20 0.46
PTPN1 P18031 4/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
ESR1 P03372 2/20 0.41
CYP1A1 P04798 2/20 0.40
CYP1B1 Q16678 2/20 0.40
DPP4 P27487 1/20 0.40
ESRRG P62508 1/20 0.40
P4HB P07237 2/20 0.40
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852544 0.90 KDM4E (0.47) KDM4ESNCAPTPN1CYP1A1CYP1B1
SCHEMBL4853546 0.87 SNCA (0.48) KDM4ESNCAPTPN1BCHEACHE
SCHEMBL4849762 0.87 KDM4E (0.52) KDM4EPTPN1BCHEACHECYP1A1
SCHEMBL4847320 0.83 SNCA (0.44) SNCAPTPN1BCHEACHEDPP4
SCHEMBL4856299 0.82 MCL1 (0.50) KDM4ESNCABCHEACHEESR1
SCHEMBL4854973 0.82 MCL1 (0.50) KDM4ESNCABCHEACHEESR1
SCHEMBL4850027 0.80 TNFRSF1A (0.47) KDM4ESNCAPTPN1BCHEACHE
SCHEMBL4847397 0.79 LMNA (0.49) KDM4EPTPN1CYP1A1CYP1B1GAA
SCHEMBL4854287 0.77 PTPN1 (0.55) PTPN1BCHEACHECYP1A1CYP1B1
SCHEMBL5915428 0.77 PTPN1 (0.53) SNCAPTPN1CYP1A1CYP1B1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed