SCHEMBL4858562

SCHEMBL4858562

[c]1cccc(NCc2ccncc2)c1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 2/20 0.49
HTT P42858 2/20 0.44
ADRA2C P18825 1/20 0.44
GAA P10253 2/20 0.42
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
ALDH1A1 P00352 1/20 0.42
PABPC1 P11940 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
RAB9A P51151 1/20 0.41
LTA4H P09960 1/20 0.41
F2 P00734 3/20 0.41
ALOX12 P18054 1/20 0.41
CA9 Q16790 1/20 0.41
PRSS1 P07477 1/20 0.39
MAPKAPK2 P49137 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL698363 0.84 HTT (0.48) KCNH3HTTKDM4EMAPTALDH1A1
SCHEMBL522061 0.77 KCNH3 (0.68) KCNH3HTTADRA2CLTA4HF2
SCHEMBL1043672 0.77 SLC2A4 (0.51) HTTGAAMAPTALDH1A1NPSR1
SCHEMBL3318487 0.76 LTA4H (0.57) GAAKDM4EMAPTALDH1A1PABPC1
SCHEMBL19241691 0.75 F2 (0.56) KCNH3HTTADRA2CGAAKDM4E
SCHEMBL19242049 0.75 KDM4E (0.61) KCNH3HTTADRA2CGAAKDM4E
SCHEMBL28330956 0.74 F2 (0.49) KCNH3HTTADRA2CGAAKDM4E
SCHEMBL2526849 0.74 RAD52 (0.45) KCNH3ADRA2CKDM4EMAPTALDH1A1
SCHEMBL19242051 0.71 F2 (0.61) KCNH3HTTGAAKDM4EMAPT
SCHEMBL1451843 0.71 CYP11B1 (0.41) MAPTLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465900-B1 RHO-KINASE INHIBITORS BAYER HEALTHCARE AG (DE) 2008-05-14 EP claimed