SCHEMBL485983

SCHEMBL485983

CC1(C)CC(Nc2ccccc2Cl)c2cc(C(=O)O)ccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
LMNA P02545 1/20 0.41
PTK2B Q14289 2/20 0.40
KDM4E B2RXH2 2/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
RXRA P19793 5/20 0.38
P2RX7 Q99572 1/20 0.38
SLC6A4 P31645 2/20 0.38
PPARG P37231 1/20 0.38
NR1H4 Q96RI1 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
RARB P10826 4/20 0.38
RARG P13631 4/20 0.38
PYGL P06737 2/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15235436 0.83 PYGL (0.46) NPC1RAB9AALDH1A1RXRAP2RX7
SCHEMBL485985 0.83 PYGL (0.46) NPC1RAB9AALDH1A1RXRAP2RX7
SCHEMBL878046 0.73 SMN1; SMN2 (0.45) SMN1; SMN2NPC1RAB9ALMNAPTK2B
SCHEMBL1071564 0.72 RXRA (0.46) RXRARARBRARGCYP26A1RARA
SCHEMBL803655 0.71 RXRA (0.41) TSHRALDH1A1MAPTRXRARARB
SCHEMBL13189905 0.71 KDM1A (0.46) RXRARARBRARGCYP26A1RARA
SCHEMBL27915456 0.65 MAPT (0.51) SMN1; SMN2NPC1RAB9ALMNAPTK2B
SCHEMBL2815476 0.64 PYGL (0.46) NPC1RAB9AALDH1A1P2RX7SLC6A4
SCHEMBL17276229 0.64 NPC1 (0.42) SMN1; SMN2NPC1RAB9ATSHRALDH1A1
SCHEMBL23362424 0.64 CNR1 (0.41) RXRARARBRARGTRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411381-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-02-01 EP disclosed
WO-2010108651-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2010-09-30 WO disclosed