SCHEMBL878046

SCHEMBL878046

O=C(O)c1ccc2c(c1)CCC2Nc1ccccc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
RAB9A P51151 1/20 0.45
TAS1R3 Q7RTX0 5/20 0.45
TAS1R1 Q7RTX1 5/20 0.45
PTK2B Q14289 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TSHR P16473 1/20 0.44
TAS1R2 Q8TE23 3/20 0.44
FADS1 O60427 1/20 0.43
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
PYGL P06737 1/20 0.40
PYGM P11217 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
SRD5A1 P18405 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL785412 0.81 TAS1R3 (0.62) TAS1R3TAS1R1TAS1R2ALDH1A1PYGL
SCHEMBL878113 0.81 TAS1R3 (0.40) SMN1; SMN2TAS1R3TAS1R1PTK2BTSHR
SCHEMBL785296 0.81 TAS1R3 (0.62) TAS1R3TAS1R1TAS1R2ALDH1A1PYGL
SCHEMBL2815355 0.81 TAS1R3 (0.62) TAS1R3TAS1R1TAS1R2ALDH1A1PYGL
SCHEMBL784591 0.79 CYP1A2 (0.50) SMN1; SMN2TAS1R3TAS1R1PTK2BKDM4E
SCHEMBL786013 0.79 CYP1A2 (0.50) SMN1; SMN2TAS1R3TAS1R1PTK2BKDM4E
SCHEMBL8181063 0.78 ALDH1A1 (0.45) TAS1R3TAS1R1KDM4ETAS1R2ALDH1A1
SCHEMBL8255449 0.76 PDPK1 (0.51) TAS1R3TAS1R1KDM4EALDH1A1MAPT
SCHEMBL10405757 0.73 CYP1A2 (0.65) SMN1; SMN2TSHRALDH1A1PDE4APDE4B
SCHEMBL485983 0.73 SMN1; SMN2 (0.41) SMN1; SMN2NPC1LMNARAB9APTK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619178-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2013-07-31 EP disclosed
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed