SCHEMBL4859932

SCHEMBL4859932

CN1C(=O)SC(CC(N)=O)C1=O

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.49
GAA P10253 5/20 0.49
KDM4E B2RXH2 4/20 0.49
NPC1 O15118 1/20 0.49
GLA P06280 1/20 0.49
HPGD P15428 3/20 0.43
RECQL P46063 1/20 0.43
POLB P06746 1/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
MAPT P10636 2/20 0.35
HSD17B10 Q99714 1/20 0.34
THRB P10828 1/20 0.33
LMNA P02545 1/20 0.33
ADAM17 P78536 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23346814 0.65
SCHEMBL7459354 0.62
SCHEMBL10686440 0.60
SCHEMBL18884239 0.57 ALDH1A1 (0.38) ALDH1A1GAAKDM4EHPGDPOLB
SCHEMBL20374229 0.57 ALDH1A1 (0.38) ALDH1A1GAAKDM4EHPGDPOLB
SCHEMBL26273902 0.55
SCHEMBL1618636 0.55
SCHEMBL17294238 0.52
Propionamide SCHEMBL11420245 0.50 TDP1 (0.47) ALDH1A1KDM4EGLAHPGDRECQL
Propionamide SCHEMBL11420169 0.50 TDP1 (0.47) ALDH1A1KDM4EGLAHPGDRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008099165-A1 PIPERIDINE DERIVATIVES AND THEIR USE FOR TREATMENT OF CCR8 MEDIATED DISEASES ASTRAZENECA AB (SE) 2008-08-21 WO disclosed