SCHEMBL4860205

SCHEMBL4860205

CCCc1c(C(=O)C(=O)C2=C(Cc3ccccc3F)N(N3CCC(c4cn(Cc5ccccc5F)c5ccccc45)C3)N(c3ccccc3)C2CCC)cnn1-c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
NOD2 Q9HC29 1/20 0.34
LMNA P02545 1/20 0.34
ALOX12 P18054 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 4/20 0.33
HRH2 P25021 3/20 0.33
MAPK1 P28482 3/20 0.32
MAPK14 Q16539 1/20 0.32
GAA P10253 1/20 0.32
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852957 0.81 ALDH1A1 (0.44) ALDH1A1NPC1RAB9ANOD2LMNA
SCHEMBL773204 0.59 NR4A3 (0.78) ALDH1A1LMNAPOLBMAPTMAPK1
SCHEMBL5206324 0.57 SLC2A1 (0.50) ALDH1A1LMNAHTTNPSR1POLB
SCHEMBL16615597 0.57 ALDH1A1 (0.74) ALDH1A1LMNANPSR1MAPTMAPK1
SCHEMBL13593554 0.56 ALDH1A1 (0.63) ALDH1A1LMNAPOLBMAPTMAPK1
SCHEMBL4851314 0.56 HTR6 (0.45) ALDH1A1NPC1RAB9ANOD2LMNA
SCHEMBL27808 0.56 NR4A3 (0.61) ALDH1A1LMNAPOLBMAPTMAPK1
SCHEMBL14927230 0.56 RAB9A (0.78) ALDH1A1NPC1RAB9ANOD2LMNA
SCHEMBL1549166 0.56 MAPT (0.76) ALDH1A1NPC1RAB9ANOD2LMNA
SCHEMBL2857718 0.56 ALDH1A1 (0.69) ALDH1A1LMNAPOLBMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7368470-B2 Substituted 3-pyrrolidine-indole derivatives GRUENENTHAL GMBH (DE) 2008-05-06 US disclosed