SCHEMBL4861660

SCHEMBL4861660

[O]c1ccc(CC2C(=O)NOC2=O)cc1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.34
GLA P06280 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
GSK3B P49841 1/20 0.33
MAPT P10636 2/20 0.31
KDM4E B2RXH2 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16520282 0.84 GAA (0.40) GAAGLANPSR1MAPTKDM4E
SCHEMBL4861014 0.66
SCHEMBL14217545 0.66
SCHEMBL5522518 0.60 MGLL (0.33) GAA
SCHEMBL13399578 0.55 MDM2 (0.47) KDM4E
SCHEMBL18751777 0.54 HDAC8 (0.56) GAA
SCHEMBL10767764 0.54 IDO1 (0.33) NPSR1GSK3BMAPT
SCHEMBL17717914 0.51 ALDH1A1 (0.72) GAAMAPTKDM4EL3MBTL1
SCHEMBL7191433 0.48 PANK3 (0.32)
SCHEMBL4398792 0.48 ESR1 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7355054-B2 Indole derivatives NEURIM PHARMACEUTICALS (1991) LTD. (IL) 2008-04-08 US claimed
US-20050159463-A1 Indole derivatives NEURIM PHARMACEUTICALS (1991) LTD. (IL) 2005-07-21 US claimed
EP-1189583-B1 INDOLE DERIVATIVES NEURIM PHARMA 1991 (IL) 2005-07-20 EP claimed
EP-1189583-A4 INDOLE DERIVATIVES NEURIM PHARMA 1991 (IL) 2004-04-14 EP claimed
EP-1189583-A1 INDOLE DERIVATIVES NEURIM PHARMACEUTICALS (1991) LIMITED (IL) 2002-03-27 EP claimed
WO-2000072815-A1 INDOLE DERIVATIVES NEURIM PHARMACEUTICALS (1991) LTD. (IL) 2000-12-07 WO claimed
US-7355054-B2 Indole derivatives NEURIM PHARMACEUTICALS (1991) LTD. (IL) 2008-04-08 US disclosed
US-20050159463-A1 Indole derivatives NEURIM PHARMACEUTICALS (1991) LTD. (IL) 2005-07-21 US disclosed
EP-1189583-B1 INDOLE DERIVATIVES NEURIM PHARMA 1991 (IL) 2005-07-20 EP disclosed
US-6858642-B1 Indole derivatives NEURIM PHARMACEUTICALS (1991) LTD. (IL) 2005-02-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050159463-A1 Indole derivatives IDO1, IDO2, H1-0 GAA 3833/4885GLA 197/4885NPSR1 438/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.