SCHEMBL4866880

SCHEMBL4866880

CN(C)S(=O)(=O)N[C@@H](Cc1cc[c]cc1)C(=O)NCCCCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
AVPR1B P47901 1/20 0.44
MMP8 P22894 1/20 0.44
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
NPY5R Q15761 1/20 0.42
PTPN1 P18031 2/20 0.42
REN P00797 1/20 0.42
CNR1 P21554 1/20 0.42
KDM4A O75164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4866881 1.00 KMT2A (0.45) KMT2ACYP2D6CYP2C9CYP2C19AVPR1B
SCHEMBL4864204 0.86 KMT2A (0.49) KMT2ACYP2D6CYP2C9CYP2C19MMP8
SCHEMBL4864202 0.86 KMT2A (0.49) KMT2ACYP2D6CYP2C9CYP2C19MMP8
SCHEMBL4857259 0.83 NPY5R (0.62) ALDH1A1NPY5R
SCHEMBL4857262 0.83 NPY5R (0.62) ALDH1A1NPY5R
SCHEMBL4866934 0.82 GRIA1 (0.46) KMT2ACYP2D6CYP2C9CYP2C19MMP8
SCHEMBL4866943 0.82 GRIA1 (0.46) KMT2ACYP2D6CYP2C9CYP2C19MMP8
SCHEMBL3738289 0.82 PTPN1 (0.48) AVPR1BPTPN1
SCHEMBL3738292 0.82 PTPN1 (0.48) AVPR1BPTPN1
SCHEMBL4858174 0.81 MMP2 (0.56) ALDH1A1NPY5RCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008520575-A 2008-06-19 JP claimed
EP-1812012-A2 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Ceptyr, Inc. (US) 2007-08-01 EP claimed
WO-2006055525-A2 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF CEPTYR, INC. (US) 2006-05-26 WO claimed
EP-1812012-A2 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Ceptyr, Inc. (US) 2007-08-01 EP disclosed
WO-2006055525-A2 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF CEPTYR, INC. (US) 2006-05-26 WO disclosed