SCHEMBL4867147

SCHEMBL4867147

O=C(O)c1c(-c2ccc(C(F)(F)F)cc2)nn2cccnc12

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 4/20 0.52
KCNQ2 O43526 4/20 0.52
JAK2 O60674 1/20 0.41
PTGS2 P35354 1/20 0.41
PPARG P37231 1/20 0.41
RORC P51449 1/20 0.41
TRPV1 Q8NER1 5/20 0.40
DHODH Q02127 2/20 0.40
SLC6A7 Q99884 1/20 0.39
PTGER1 P34995 1/20 0.38
TLR7 Q9NYK1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3175267 0.87 KMO (0.46) KCNQ3KCNQ2PTGS2DHODHSLC6A7
SCHEMBL14710420 0.83 PTGS2 (0.41) KCNQ3KCNQ2PTGS2RORCTRPV1
SCHEMBL29939968 0.80 HTR6 (0.43) KCNQ3KCNQ2JAK2PTGS2RORC
SCHEMBL30627413 0.77 ELANE (0.42) KCNQ3KCNQ2PPARGRORC
SCHEMBL23023568 0.75 PTGS2 (0.41) KCNQ3KCNQ2PTGS2RORC
SCHEMBL15210509 0.75 POLB (0.48) KCNQ3KCNQ2PTGS2
SCHEMBL27230023 0.75 PIK3CD (0.46) KCNQ3KCNQ2JAK2
SCHEMBL29703839 0.74 DHODH (0.42) PTGS2DHODH
SCHEMBL23013809 0.74 DHODH (0.42) PTGS2DHODH
SCHEMBL30028953 0.74 KCNQ3 (0.38) KCNQ3KCNQ2PTGS2PPARGRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008530042-A 2008-08-07 JP claimed
EP-1851225-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. Hoffmann-Roche AG (CH) 2007-11-07 EP claimed
WO-2006084634-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2006-08-17 WO claimed