SCHEMBL4868324

SCHEMBL4868324

CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)C(CO)NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.48
HRH2 P25021 2/20 0.41
HRH1 P35367 2/20 0.41
SCN9A Q15858 3/20 0.41
CYP3A4 P08684 1/20 0.41
RAB9A P51151 1/20 0.39
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
PTPN1 P18031 2/20 0.38
SSTR1 P30872 1/20 0.38
SSTR4 P31391 1/20 0.38
EPHX2 P34913 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4871244 0.90 HRH2 (0.41) HRH2HRH1SCN9ARAB9AHDAC4
SCHEMBL4871968 0.89 AVPR1A (0.44) HRH2HRH1RAB9AHDAC4HDAC1
SCHEMBL4865092 0.85 HRH2 (0.44) HRH2HRH1SCN9ARAB9AHDAC4
SCHEMBL4868460 0.83 AVPR1A (0.50) CTSLSCN9A
SCHEMBL4865061 0.82 SCN9A (0.49) CTSLSCN9A
SCHEMBL4868278 0.82 SCN9A (0.53) CTSLSCN9A
SCHEMBL4873124 0.81 CTSS (0.55) CTSLSCN9A
SCHEMBL4861830 0.79 SUV39H2 (0.43) SCN9AHDAC4HDAC1HDAC6
SCHEMBL4864055 0.79 SCN9A (0.49) CTSLSCN9A
SCHEMBL4861770 0.78 SCN9A (0.50) CTSLSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751090-B1 ACID DERIVATIVES OF SUBSTITUTED CYCLOHEXYL-1,4-DIAMINES GRUENENTHAL GMBH (DE) 2014-10-08 EP claimed
US-7439394-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2008-10-21 US claimed
US-20070117803-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-24 US claimed
EP-1751090-B1 ACID DERIVATIVES OF SUBSTITUTED CYCLOHEXYL-1,4-DIAMINES GRUENENTHAL GMBH (DE) 2014-10-08 EP disclosed
US-7439394-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2008-10-21 US disclosed
US-20070117803-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070117803-A1 Cyclohexyl-1,4-diamine compounds PKD1, DDC, DPYD CTSL 2008/4885HRH2 181/4885HRH1 121/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.