SCHEMBL4871968

SCHEMBL4871968

CN(C)C1(Cc2ccc(Cl)cc2)CCC(NC(=O)C(CO)NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 10/20 0.44
CACNA1B Q00975 1/20 0.44
HRH2 P25021 2/20 0.43
HRH1 P35367 2/20 0.43
OXTR P30559 1/20 0.42
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KCNH2 Q12809 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4865092 0.92 HRH2 (0.44) CACNA1BHRH2HRH1PPARGPPARA
SCHEMBL4868460 0.89 AVPR1A (0.50) AVPR1AOXTR
SCHEMBL4868324 0.89 CTSL (0.48) HRH2HRH1HDAC4HDAC1HDAC6
SCHEMBL4861830 0.89 SUV39H2 (0.43) AVPR1ACACNA1BOXTRPPARGPPARA
SCHEMBL4871244 0.85 HRH2 (0.41) HRH2HRH1HDAC4HDAC1HDAC6
SCHEMBL4868278 0.83 SCN9A (0.53)
SCHEMBL4861770 0.81 SCN9A (0.50)
SCHEMBL4864032 0.79 DRD2 (0.44)
SCHEMBL4864055 0.78 SCN9A (0.49)
SCHEMBL4865061 0.76 SCN9A (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439394-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2008-10-21 US claimed
US-20070117803-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-24 US claimed
EP-1751090-B1 ACID DERIVATIVES OF SUBSTITUTED CYCLOHEXYL-1,4-DIAMINES GRUENENTHAL GMBH (DE) 2014-10-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070117803-A1 Cyclohexyl-1,4-diamine compounds PKD1, DDC, DPYD AVPR1A 2695/4885CACNA1B 3036/4885HRH2 181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.