SCHEMBL4868657

SCHEMBL4868657

NC(=O)CCC(CP(=O)(O)Cc1ccc(F)cc1)C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.51
GRM3 Q14832 2/20 0.45
MMP1 P03956 2/20 0.44
MMP13 P45452 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5053155 0.89 FOLH1 (0.64) FOLH1GRM3
SCHEMBL4873564 0.86 FOLH1 (0.45) FOLH1GRM3MMP1MMP13
SCHEMBL14112042 0.80 FOLH1 (0.42) FOLH1GRM3
SCHEMBL14112041 0.80 FOLH1 (0.79) FOLH1GRM3
SCHEMBL6682065 0.78 MMP1 (0.46) FOLH1MMP1
SCHEMBL12628838 0.77 GRM3 (0.61) FOLH1GRM3
SCHEMBL4874698 0.77 FOLH1 (0.39) FOLH1GRM3
SCHEMBL1373664 0.76 GRM3 (0.65) FOLH1GRM3
SCHEMBL4874207 0.76 CYP26B1 (0.44) FOLH1
SCHEMBL5051119 0.76 GRM3 (0.59) FOLH1GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7402576-B2 Phosphinic acid analogs of glutamate GIVAUDAN SA (CH) 2008-07-22 US disclosed
US-7402576-B2 Phosphinic acid analogs of glutamate GIVAUDAN SA (CH) 2008-07-22 US disclosed
US-7402576-B2 Phosphinic acid analogs of glutamate GIVAUDAN SA (CH) 2008-07-22 US disclosed
EP-1599487-B1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE GIVAUDAN SA (CH) 2007-07-11 EP disclosed
EP-1599487-B1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE GIVAUDAN SA (CH) 2007-07-11 EP disclosed
US-20060052616-A1 Phosphinic acid analogs of glutamate GIVAUDAN SA (CH) 2006-03-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052616-A1 Phosphinic acid analogs of glutamate GLUL, GRIA1, GRM1 FOLH1 70/4885GRM3 35/4885MMP1 4142/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.