SCHEMBL4868911

SCHEMBL4868911

NC(=O)CCC(C(=O)O)C(O)(C/C=C/c1ccccc1)P=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 4/20 0.38
GRIK2 Q13002 3/20 0.38
PAM P19021 1/20 0.37
KMT2A Q03164 1/20 0.33
MMP2 P08253 2/20 0.33
MMP9 P14780 2/20 0.33
HTR2A P28223 3/20 0.33
HTT P42858 1/20 0.33
MAOB P27338 1/20 0.33
CYP1A2 P05177 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4868908 0.81 GRIK1 (0.38) GRIK1GRIK2PAMKMT2AMMP9
SCHEMBL4868913 0.81 GRIK1 (0.38) GRIK1GRIK2PAMKMT2AMMP9
SCHEMBL3514739 0.76 ALOX15 (0.37) KMT2AHTT
SCHEMBL4874792 0.74 GRIK1 (0.39) GRIK1
SCHEMBL4865814 0.73 MAPT (0.39) GRIK1
SCHEMBL4868970 0.72 KMT2A (0.43) KMT2AMMP2MMP9
SCHEMBL6682070 0.71 GGPS1 (0.45) KMT2AMMP2MMP9
SCHEMBL4871624 0.71 SLC1A3 (0.39) CYP1A2
SCHEMBL4869123 0.71 TSHR (0.36) KMT2AHTTCYP1A2ALDH1A1
SCHEMBL4868669 0.70 KIF11 (0.35) KMT2AMMP2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7402576-B2 Phosphinic acid analogs of glutamate GIVAUDAN SA (CH) 2008-07-22 US disclosed
EP-1599487-B1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE GIVAUDAN SA (CH) 2007-07-11 EP disclosed
US-20060052616-A1 Phosphinic acid analogs of glutamate GIVAUDAN SA (CH) 2006-03-09 US disclosed
EP-1599487-A1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE Givaudan SA (CH) 2005-11-30 EP disclosed
WO-2004043971-A1 PHOSPHINIC ACID ANALOGS OF GLUTAMATE GIVAUDAN SA (CH) 2004-05-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052616-A1 Phosphinic acid analogs of glutamate GLUL, GRIA1, GRM1 GRIK1 22/4885GRIK2 58/4885PAM 1031/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.