SCHEMBL4870608

SCHEMBL4870608

CC(S)S.[AsH2]c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
TAAR1 Q96RJ0 4/20 0.33
SLC6A2 P23975 3/20 0.33
LMNA P02545 3/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
MAOA P21397 1/20 0.33
TSHR P16473 1/20 0.33
ALOX12 P18054 1/20 0.33
ACHE P22303 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
CYP2A6 P11509 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
ADRA2A P08913 2/20 0.32
CYP2D6 P10635 2/20 0.32
CHRM2 P08172 1/20 0.32
HTR1A P08908 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL456859 0.80
Bromide SCHEMBL11113762 0.77
Bromide SCHEMBL28610589 0.77
Water SCHEMBL28363985 0.77
SCHEMBL9438540 0.77
Biphenyl SCHEMBL11779724 0.69 ALDH1A1 (0.60) TDP1TAAR1SLC6A4CYP1A2CYP3A4
Phenol SCHEMBL20741797 0.69 CA12 (0.61) TDP1TSHRCYP3A4
Anisole SCHEMBL11110211 0.67 CA4 (0.74) LMNATSHRACHECYP2A6DRD3
SCHEMBL664987 0.67
SCHEMBL184638 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7381572-B2 Reagents and procedures for multi-label high-specificity labeling RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2008-06-03 US disclosed
US-7282373-B2 Ultra-high specificity fluorescent labeling RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2007-10-16 US disclosed
US-7141655-B2 Reagents and procedures for high-specificity labeling RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2006-11-28 US disclosed
US-20060141531-A1 Ultra-high specificity fluorescent labeling RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2006-06-29 US disclosed
US-20060141530-A1 Using arsenic-mediated labeling to permit orthogonal molecule-specific, site-specific labeling of target molecules, such as proteins, with multiple labels; complex of peptide with tag of a cyanine dye having pendant 2,5-dithia-arsacyclopentane groups RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2006-06-29 US disclosed
US-20040019104-A1 Reagents and procedures for high-specificity labeling RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2004-01-29 US disclosed
WO-2003107010-A1 REAGENTS AND PROCEDURES FOR HIGH-SPECIFICITY LABELING RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2003-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060141531-A1 Ultra-high specificity fluorescent labeling RPS27A, RAET1L, QRFPR TDP1 2886/4885TAAR1 1582/4885SLC6A2 2685/4885
US-20060141530-A1 Using arsenic-mediated labeling to permit orthogonal molecule-specific, site-specific labeling of target molecules, such as proteins, with multiple labels; complex of peptide with tag of a cyanine dye having pendant 2,5-dithia-arsacyclopentane groups AS3MT, ARSA, PTMS TDP1 722/4885TAAR1 401/4885SLC6A2 1548/4885
US-20040019104-A1 Reagents and procedures for high-specificity labeling AS3MT, SRMS, HNRNPH3 TDP1 908/4885TAAR1 179/4885SLC6A2 729/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.