SCHEMBL4882593

SCHEMBL4882593

NN(C(=O)c1ccc2c(c1)OCO2)c1nc2c(s1)Cc1ccccc1-2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.44
CHEK1 O14757 1/20 0.42
DAPK3 O43293 1/20 0.42
LTK P29376 1/20 0.42
MAPK8 P45983 1/20 0.42
CSNK1A1 P48729 1/20 0.42
CDK8 P49336 1/20 0.42
LIMK1 P53667 1/20 0.42
CDK5 Q00535 1/20 0.42
DYRK1A Q13627 1/20 0.42
LRRK2 Q5S007 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
HPGD P15428 4/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 5/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3340579 0.76 MAPT (0.51) ADORA1HPGDNPC1RAB9AALDH1A1
SCHEMBL4801840 0.73 CHEK1 (0.43) ADORA1CHEK1DAPK3LTKMAPK8
SCHEMBL4799024 0.71 KMT2A (0.53) ADORA1HPGDNPC1RAB9AALDH1A1
SCHEMBL7863728 0.70 ALDH1A1 (0.60) HPGDNPC1RAB9AALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL11829820 0.69 ALDH1A1 (0.58) HPGDNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL4882626 0.67 HPGD (0.38) HPGDNPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL4959981 0.64 CHEK1 (0.60) ADORA1CHEK1DAPK3LTKMAPK8
SCHEMBL4799172 0.63 MAPT (0.49) NPC1RAB9AALDH1A1SMN1; SMN2MEN1
SCHEMBL13943068 0.63 ADORA1 (0.98) ADORA1
SCHEMBL31151793 0.61 HPGD (0.65) HPGDNPC1RAB9AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052804-A1 THIAZOLHYDRAZIDES FOR TREATMENT OF NEURODEGENERATIVE DISEASES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2008-05-08 WO disclosed