SCHEMBL4884759

SCHEMBL4884759

CCCCCS[C@@]1(n2cnc3c(N)ncnc32)O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EHMT1 Q9H9B1 1/20 0.48
PI4KA P42356 2/20 0.46
PI4K2B Q8TCG2 2/20 0.46
PI4K2A Q9BTU6 2/20 0.46
PI4KB Q9UBF8 2/20 0.46
ADORA3 P0DMS8 5/20 0.45
ADORA2A P29274 5/20 0.45
ADORA2B P29275 3/20 0.45
SLC28A1 O00337 2/20 0.45
DPP4 P27487 1/20 0.45
MEN1 O00255 1/20 0.45
MAP3K7 O43318 1/20 0.45
SLC28A2 O43868 1/20 0.45
GAPDH P04406 1/20 0.45
MAPK1 P28482 1/20 0.45
ADORA1 P30542 1/20 0.45
STAT6 P42226 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
DOT1L Q8TEK3 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL998090 0.90 PI4KA (0.48) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL30216733 0.86 EHMT1 (0.45) EHMT1ADORA3ADORA2ASLC28A1GMPS
SCHEMBL160357 0.86 ADORA3 (0.53) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL9495963 0.85 PI4KA (0.46) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL28160452 0.84 ADORA3 (0.45) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL6935380 0.83 PI4KA (0.48) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL9231750 0.82 ADORA3 (0.49) EHMT1PI4KAPI4K2BPI4K2API4KB
SCHEMBL5742060 0.82 PI4KA (0.47) PI4KAPI4K2BPI4K2API4KBADORA3
SCHEMBL3317153 0.82 ADORA2A (0.48) EHMT1PI4KAPI4K2BPI4K2API4KB
SCHEMBL1920532 0.81 ADORA3 (0.48) EHMT1PI4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7348315-B2 Methods of treating heart failure with modified ATP, ADP and AMP compounds THE UNIVERSITY OF CONNECTICUT (US) 2008-03-25 US disclosed
US-20030186929-A1 Methods of treating heart failure with modified ATP, ADP and AMP compounds NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2003-10-02 US disclosed
US-6255292-B1 INCREASING CELLULAR CONTRACTIONS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA 2001-07-03 US disclosed
US-5712258-A Inotropic ADP and ATP analogues and their pharmaceutical compositions THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1998-01-27 US disclosed
WO-1996029345-A1 NOVEL INOTROPIC AGENTS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 1996-09-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030186929-A1 Methods of treating heart failure with modified ATP, ADP and AMP compounds ATP5MF, ATP5MG, ATP2A1 EHMT1 1868/4885PI4KA 2498/4885PI4K2B 3654/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.