SCHEMBL4885149

SCHEMBL4885149

CC(C)C1CCC(C)(CCl)CC1O

nearest known ligand 0.36

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.36
TRPM8 Q7Z2W7 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8088736 1.00 TRPA1 (0.36) TRPA1TRPM8
SCHEMBL8183428 1.00 TRPA1 (0.36) TRPA1TRPM8
SCHEMBL3269762 0.84 TRPA1 (0.37) TRPA1TRPM8
SCHEMBL584356 0.84 TRPA1 (0.37) TRPA1TRPM8
SCHEMBL5926940 0.84 TRPA1 (0.37) TRPA1TRPM8
SCHEMBL6907615 0.84 TRPA1 (0.37) TRPA1TRPM8
SCHEMBL27824250 0.82 TRPA1 (0.36) TRPA1TRPM8
SCHEMBL27488960 0.81 TRPA1 (0.35) TRPA1TRPM8
SCHEMBL28317324 0.81 TRPA1 (0.35) TRPA1TRPM8
SCHEMBL4733415 0.81 TRPA1 (0.35) TRPA1TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080132689-A1 Complexing using an ortho carboxy acetal; biodrug delivery ROCHE MADISON INC 2008-06-05 US disclosed
US-7348453-B2 Labile linkage for compound delivery to a cell MIRUS BIO CORPORATION (US) 2008-03-25 US disclosed
WO-2005026253-A2 LABILE LINKAGE FOR COMPOUND DELIVERY TO A CELL MIRUS BIO CORPORATION (US) 2005-03-24 WO disclosed
US-20050054604-A1 Labile linkage for compound delivery to a cell ROCHE MADISON INC. 2005-03-10 US disclosed
US-6162932-A Stereoselective synthesis of endothelin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2000-12-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050054604-A1 Labile linkage for compound delivery to a cell AADAC, PAICS, FURIN TRPA1 3803/4885TRPM8 3152/4885
US-20080132689-A1 Complexing using an ortho carboxy acetal; biodrug delivery CEL, PAICS, OGA TRPA1 4058/4885TRPM8 4056/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.