Glisoxepide

Glisoxepide

SCHEMBL48892

Cc1cc(C(=O)NCCc2ccc(S(=O)(=O)NC(=O)NN3CCCCCC3)cc2)no1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.55
ALDH1A1 P00352 5/20 0.54
MAPT P10636 4/20 0.54
CYP3A4 P08684 3/20 0.54
NFKB1 P19838 2/20 0.54
TP53 P04637 2/20 0.54
KDM4E B2RXH2 1/20 0.54
GLA P06280 1/20 0.54
GAA P10253 1/20 0.54
ALOX12 P18054 1/20 0.54
CYP2C9 P11712 2/20 0.51
TSHR P16473 2/20 0.51
CYP2C19 P33261 2/20 0.51
BLM P54132 2/20 0.51
HTR1A P08908 1/20 0.51
CNR1 P21554 1/20 0.51
ADRA1A P35348 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
POLB P06746 2/20 0.46
CA12 O43570 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Glisolamide SCHEMBL27735549 0.90 CYP3A4 (0.62) LMNAALDH1A1MAPTCYP3A4NFKB1
SCHEMBL23893971 0.89 LMNA (0.53) LMNAALDH1A1MAPTCYP3A4NFKB1
Glisoxepide SCHEMBL28142826 0.86 LMNA (0.57) LMNAALDH1A1MAPTCYP3A4NFKB1
Glisolamide SCHEMBL38106 0.84 LMNA (0.73) LMNAALDH1A1MAPTCYP3A4NFKB1
SCHEMBL11630344 0.81 ALDH1A1 (0.63) LMNAALDH1A1MAPTCYP3A4NFKB1
Glimepiride SCHEMBL28086735 0.80 CYP2C9 (0.72) LMNAALDH1A1MAPTCYP3A4NFKB1
SCHEMBL11628147 0.80 ALDH1A1 (0.53) LMNAALDH1A1MAPTCYP3A4NFKB1
SCHEMBL18007638 0.80 NLRP3 (0.58) LMNANLRP3
SCHEMBL11627816 0.80 MAPT (0.57) LMNAALDH1A1MAPTCYP3A4NFKB1
SCHEMBL11624368 0.79 ALDH1A1 (0.53) LMNAALDH1A1MAPTCYP3A4NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4356 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4640701-A2 GLUCAGON LIKE PEPTIDE 1 (GLP-1) FUSION PEPTIDE COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE CONJUGATES AND USES THEREOF Janssen Sciences Ireland Unlimited Company (IE) 2025-10-29 EP claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-4520343-A2 GLUCAGON LIKE PEPTIDE 1 (GLP1)-GROWTH DIFFERENTIATION FACTOR 15 (GDF15) FUSION PROTEINS AND USES THEREOF Janssen Sciences Ireland Unlimited Company (IE) 2025-03-12 EP claimed
EP-3988123-B1 ANTIBODY-COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODULATORS OF NEUROPEPTIDE Y RECEPTORS JANSSEN PHARMACEUTICA NV (BE) 2025-02-26 EP claimed
US-12208071-B2 Glucagon receptor antagonists LIGAND PHARMACEUTICALS INCORPORATED (US) 2025-01-28 US claimed
US-12186329-B2 Compositions and methods related to cholic acid 7-sulfate as a treatment for diabetes PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2025-01-07 US claimed
US-20240366579-A1 PHARMACEUTICAL COMPOSITION COMPRISING GPR40 AGONIST AND SGLT-2 INHIBITOR ILDONG PHARMACEUTICAL CO., LTD. (KR) 2024-11-07 US claimed
US-20240316048-A1 Prevention of Pancreatic Cell Degeneration MELIOR PHARMACEUTICALS I, INC. 2024-09-26 US claimed
US-12070461-B2 Methods and formulations for modulating Lyn kinase activity and treating related disorders MELIOR PHARMACEUTICALS I, INC. (US) 2024-08-27 US claimed
EP-4329756-A1 PHARMACEUTICAL COMPOSITION COMPRISING GPR40 AGONIST AND SGLT-2 INHIBITOR Ildong Pharmaceutical Co., Ltd. (KR) 2024-03-06 EP claimed
WO-1998036755-A1 SULFONYLUREA-GLITAZONE SYNERGISTIC COMBINATIONS FOR DIABETES WARNER LAMBERT COMPANY (US) 1998-08-27 WO claimed
WO-1998018610-A1 EMBEDDING AND ENCAPSULATION OF CONTROLLED RELEASE PARTICLES LENGERICH BERNHARD H VAN (US) 1998-05-07 WO claimed
CN-1170346-A Process for encapsulation of caplets in capsule and solid dasage forms obtainable by such process WARNER LAMBERT CO (US) 1998-01-14 CN claimed
WO-1997037629-A1 PROCESS FOR ENCAPSULATION OF CAPLETS IN A CAPSULE AND SOLID DOSAGE FORMS OBTAINABLE BY SUCH PROCESS WARNER-LAMBERT COMPANY (US) 1997-10-16 WO claimed
EP-0797424-A1 PROCESS FOR ENCAPSULATION OF CAPLETS IN A CAPSULE AND SOLID DOSAGE FORMS OBTAINABLE BY SUCH PROCESS WARNER-LAMBERT COMPANY (US) 1997-10-01 EP claimed
EP-0724427-A1 HIGHLY ACTIVE SULPHONYL UREA PREPARATIONS EXHIBITING RAPID OR CONTROLLED RELEASE OF THE ACTIVE SUBSTANCE, AND METHOD OF PRODUCING THEM BRITISH TECHNOLOGY GROUP LTD (GB) 1996-08-07 EP claimed
WO-1996018370-A1 PROCESS FOR ENCAPSULATION OF CAPLETS IN A CAPSULE AND SOLID DOSAGE FORMS OBTAINABLE BY SUCH PROCESS WARNER-LAMBERT COMPANY (US) 1996-06-20 WO claimed
WO-1995011006-A1 HIGHLY ACTIVE SULPHONYL UREA PREPARATIONS EXHIBITING RAPID OR CONTROLLED RELEASE OF THE ACTIVE SUBSTANCE, AND METHOD OF PRODUCING THEM BRITISH TECHNOLOGY GROUP LTD. (GB) 1995-04-27 WO claimed
US-4708868-A Oral anti-diabetic pharmaceutical forms and the preparation thereof DR. KARL THOMAE GMBH (DE) 1987-11-24 US claimed
US-4696815-A Anti-diabetic pharmaceutical forms and the preparation thereof DR. KARL THOMAE GMBH (DE) 1987-09-29 US claimed