SCHEMBL4895563

SCHEMBL4895563

CSc1cc(Cl)ccc1C[AsH2]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP1A2 P05177 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 2/20 0.39
LMNA P02545 1/20 0.39
ALDH1A1 P00352 4/20 0.36
IDO1 P14902 4/20 0.36
HPGD P15428 3/20 0.36
PLA2G1B P04054 2/20 0.36
ATG4B Q9Y4P1 2/20 0.36
HTT P42858 2/20 0.36
MEN1 O00255 1/20 0.36
HSP90AA1 P07900 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALOX15 P16050 1/20 0.36
KMT2A Q03164 1/20 0.36
HIF1A Q16665 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28167406 0.80 RAB9A (0.42) CYP3A4CYP2C9CYP2C19CYP1A2MAPK1
SCHEMBL4095951 0.80 CYP2A6 (0.41) CYP3A4CYP2C9CYP2C19CYP1A2MAPK1
SCHEMBL29070042 0.74 KEAP1 (0.46) CYP2C9ALDH1A1MAPT
SCHEMBL3787206 0.73 CCR2 (0.46) CYP3A4CYP2C9CYP2C19MAPK1RAB9A
SCHEMBL1145559 0.72 TP53 (0.48) CYP3A4CYP2C9CYP2C19CYP1A2RAB9A
SCHEMBL18850253 0.70 CCR2 (0.46) CYP3A4CYP2C9CYP2C19RAB9AALDH1A1
SCHEMBL8492853 0.70 CYP3A4 (0.48) CYP3A4CYP2C9CYP2C19RAB9AALDH1A1
SCHEMBL22411226 0.69 HPGD (0.42) CYP3A4CYP2C9CYP2C19MAPK1RAB9A
SCHEMBL30548387 0.69 HPGD (0.42) CYP3A4CYP2C9CYP2C19MAPK1RAB9A
SCHEMBL3783594 0.68 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19CYP1A2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987004-A2 SUBSTITUTED PYRIDINEAMIDE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2008-11-05 EP disclosed
WO-2007098352-A2 SUBSTITUTED PYRIDINEAMIDE COMPOUNDS USEFUL AS SOLUBLE EPOXIDE HYDROLASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-08-30 WO disclosed