SCHEMBL4900459

SCHEMBL4900459

NNC(=O)c1cnc2cnccc2c1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 10/20 0.55
KDM4E B2RXH2 2/20 0.51
MPO P05164 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2A6 P11509 1/20 0.51
CYP2C19 P33261 1/20 0.51
LRRK2 Q5S007 1/20 0.46
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ALDH1A1 P00352 1/20 0.43
P2RX7 Q99572 1/20 0.42
MGAM O43451 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CXCR4 P61073 1/20 0.41
BCAT1 P54687 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL721917 0.82 HPGDS (0.55) HPGDSKDM4EADORA3LRRK2NPC1
SCHEMBL6237473 0.81 MGAM (0.65) HPGDSKDM4ECYP1A2CYP3A4NPC1
SCHEMBL3788261 0.80 MGAM (0.64) HPGDSKDM4ELRRK2NPC1RAB9A
SCHEMBL28946126 0.78 ALOX15 (0.54) HPGDSKDM4EALDH1A1
SCHEMBL7541373 0.78 KDM4E (0.55) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL1519811 0.78 SMYD3 (0.60) KDM4EMPOCYP1A2CYP3A4ADORA3
SCHEMBL14067689 0.75 HPGDS (0.44) HPGDSKDM4ELRRK2ALDH1A1MGAM
SCHEMBL30546532 0.75 MAOB (0.56) HPGDSCYP2C19NPC1RAB9AALDH1A1
SCHEMBL1017525 0.75 MAOB (0.56) HPGDSCYP2C19NPC1RAB9AALDH1A1
Hydrochloric Acid SCHEMBL20162133 0.74 MAOB (0.55) HPGDSCYP2C19NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith D SIDOCKY NEIL R 2008-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith JAK2, CHEK2, MTOR HPGDS 111/4885KDM4E 1212/4885MPO 476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.