Sampatrilat

Sampatrilat

SCHEMBL49066

CS(=O)(=O)N[C@@H](CCCCN)C(=O)NC[C@H](CC1(C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)O)CCCC1)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 4/20 1.00
ACE P12821 3/20 1.00
MME P08473 3/20 1.00
NPPA P01160 1/20 1.00
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
ITGB1 P05556 2/20 0.39
ITGA4 P13612 2/20 0.39
CHRND Q07001 5/20 0.39
CPB2 Q96IY4 1/20 0.39
CHRNA1 P02708 1/20 0.39
CHRNG P07510 1/20 0.39
CHRNB1 P11230 1/20 0.39
MMP1 P03956 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sampatrilat SCHEMBL4567110 1.00 ECE1 (1.00) ECE1ACEMMENPPAITGB3
Sampatrilat SCHEMBL7301333 1.00 ECE1 (1.00) ECE1ACEMMENPPAITGB3
SCHEMBL7294367 0.95 ACE (0.91) ECE1ACEMMENPPAITGB3
SCHEMBL7302871 0.90 MME (0.82) ECE1ACEMMENPPAITGB3
SCHEMBL7302883 0.90 MME (0.82) ECE1ACEMMENPPAITGB3
SCHEMBL9755064 0.90 MME (0.81) ECE1ACEMMENPPAITGB1
SCHEMBL6441043 0.90 ACE (0.81) ECE1ACEMMENPPAITGB3
SCHEMBL9755065 0.90 MME (0.81) ECE1ACEMMENPPAITGB1
SCHEMBL7294361 0.89 MME (0.80) ECE1ACEMMENPPAITGB3
SCHEMBL10471733 0.88 ECE1 (0.77) ECE1ACEMMENPPAITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3724 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022265697-A1 COMPOSITIONS FOR TREATING VIRAL INFECTIONS AND METHODS FOR SAME Tiger Development, LLC (US) 2022-12-22 WO claimed
US-20220370360-A1 COMPOSITIONS FOR TREATING VIRAL INFECTIONS AND METHODS FOR SAME ACCESS TO ADVANCED HEALTH INSTITUTE 2022-11-24 US claimed
US-20210401751-A1 COMPOSITIONS FOR TREATING VIRAL INFECTIONS AND METHODS FOR SAME Tiger Development Inc. (US) 2021-12-30 US claimed
US-11166956-B2 Combinations of PDE1 inhibitors and NEP inhibitors INTRA-CELLULAR THERAPIES, INC. (US) 2021-11-09 US claimed
US-20190275046-A1 NOVEL COMBINATION INTRA-CELLULAR THERAPIES, INC. (US) 2019-09-12 US claimed
US-10285992-B2 Combinations of PDE1 inhibitors and NEP inhibitors and associated methods INTRA-CELLULAR THERAPIES, INC. (US) 2019-05-14 US claimed
US-10149909-B2 Fortifier TORAY INDUSTRIES, INC. (JP) 2018-12-11 US claimed
WO-2018211479-A1 STABILIZED COMPOSITIONS OF ANGIOTENSIN II INHIBITORS AND NEUTRAL ENDOPEPTIDASE INHIBITORS AND PROCESS FOR PREPARATION THEREOF LUPIN LIMITED (IN) 2018-11-22 WO claimed
US-10131671-B2 Organic compounds INTRA-CELLULAR THERAPIES, INC. (US) 2018-11-20 US claimed
EP-2661431-B1 HETEROCYCLIC COMPOUNDS FOR THE INHIBITION OF PASK BIOENERGENIX (US) 2018-07-11 EP claimed
US-20030065040-A1 Pharmaceutical compositions including sampatrilat dispersed in a lipoidic vehicle SUPERNUS PHARMACEUTICALS, INC 2003-04-03 US claimed
US-20030050301-A1 Combination of aldose reductase inhibitors and angiotensin-II antagonists for the treatment of diabetic nephropathy MYLARI BANAVARA L (US) 2003-03-13 US claimed
WO-2002087621-A1 PHARMACEUTICAL COMPOSITION INCLUDING ACE/NEP INHIBITORS AND BIOAVAILABILITY ENHANCERS SHIRE LABORATORIES INC. (US) 2002-11-07 WO claimed
WO-2002060437-A1 PHARMACEUTICAL COMPOSITIONS INCLUDING SAMPATRILAT DISPERSED IN A LIPOIDIC VEHICLE SHIRE LABORATORIES, INC. (US) 2002-08-08 WO claimed
WO-2002058793-A1 ESSENTIAL N-3 FATTY ACIDS IN CARDIAC INSUFFICIENCY AND HEART FAILURE THERAPY PHARMACIA ITALIA S.P.A. (IT) 2002-08-01 WO claimed
US-20020068740-A1 Combination of aldose reductase inhibitors and antihypertensive agents for the treatment of diabetic complications MYLARI BANAVARA L (US) 2002-06-06 US claimed
EP-1059918-A1 NOVEL DOSAGE FORM West Pharmaceutical Services Drug Delivery & Clinical Research Centre Limited (GB) 2000-12-20 EP claimed
WO-1999037290-A1 NOVEL DOSAGE FORM WEST PHARMACEUTICAL SERVICES DRUG DELIVERY & CLINICAL RESEARCH CENTRE LIMITED (GB) 1999-07-29 WO claimed
EP-0358398-B1 CYCLOALKYL-SUBSTITUTED GLUTARAMIDE ANTIHYPERTENSIVE AGENTS Pfizer Limited (GB) 1993-03-10 EP claimed
EP-0358398-A1 Cycloalkyl-substituted glutaramide antihypertensive agents Pfizer Limited (GB) 1990-03-14 EP claimed