Meticrane

Meticrane

SCHEMBL49070

Cc1cc2c(cc1S(N)(=O)=O)S(=O)(=O)CCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 1.00
LMNA P02545 2/20 1.00
CA2 P00918 5/20 0.46
CA1 P00915 3/20 0.44
CA9 Q16790 2/20 0.44
CYP2D6 P10635 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.33
CA12 O43570 2/20 0.33
CA7 P43166 1/20 0.33
CA14 Q9ULX7 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024678 0.91 CYP2C9 (0.83) CYP2C9LMNACA2CA1CA9
SCHEMBL11929312 0.82 LMNA (0.70) CYP2C9LMNACA2CA1CA9
SCHEMBL11925202 0.80 LMNA (0.67) CYP2C9LMNACA2KDM4EALDH1A1
Methyclothiazide SCHEMBL5886113 0.75 CHRM1 (0.71) CYP2C9LMNACA2CA1CA9
SCHEMBL6297784 0.72 CA2 (0.82) CYP2C9LMNACA2CA1CA9
SCHEMBL8030116 0.72 LMNA (0.56) CYP2C9LMNACA2CA1CA9
SCHEMBL831407 0.72 CYP2C9 (0.56) CYP2C9LMNA
SCHEMBL24871672 0.71 LMNA (0.54) CYP2C9LMNA
SCHEMBL19754398 0.69 LMNA (0.51) CYP2C9LMNACA2CA1CA9
SCHEMBL8056407 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2676 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250057876-A1 METHODS FOR TREATING AND/OR PREVENTING LYMPHANGIOGENESIS-ASSOCIATED DISEASES BY USING GOLD NANOCLUSTERS GOLDRED NANOBIOTECH CO., LTD. (TW) 2025-02-20 US claimed
US-20240009249-A1 ADIPOGENIC CELL COMPOSITIONS AND METHODS FLAGSHIP PIONEERING INNOVATIONS VI, LLC 2024-01-11 US claimed
WO-2023230770-A1 METHODS OF LUNG ADENOCARCINOMA TREATMENT WITH NON ANTI-LUAD DRUGS OR COMPOUNDS Suzhou Singleron Biotechnologies Co., Ltd. (CN) 2023-12-07 WO claimed
US-20230381161-A1 COMPOSITIONS FOR THE TREATMENT OF HYPERTENSION The George Institute for Global Health (AU) 2023-11-30 US claimed
EP-4251175-A1 ADIPOGENIC CELL COMPOSITIONS AND METHODS Flagship Pioneering, Inc. (US) 2023-10-04 EP claimed
WO-2023183932-A2 MONOBODIES BINDING TO INTERCELLULAR ADHESION MOLECULE 2 (ICAM-2) NEW YORK UNIVERSITY (US) 2023-09-28 WO claimed
WO-2023111607-A1 VALORISATION OF MARINE ANIMAL BY-PRODUCTS Goia Limited (MU) 2023-06-22 WO claimed
US-20230125076-A1 COMPOSITIONS FOR THE TREATMENT OF HYPERTENSION The George Institute for Global Health (AU) 2023-04-27 US claimed
US-20220390453-A1 OVARIAN CANCER BIOMARKER AND METHODS OF USING SAME Women's College Hospital (CA) 2022-12-08 US claimed
WO-2022115609-A1 ADIPOGENIC CELL COMPOSITIONS AND METHODS FLAGSHIP PIONEERING, INC. (US) 2022-06-02 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1086129-A1 ANTI-ANGIOGENIC PROTEINS AND METHODS OF USE THEREOF Beth Israel Deaconess Medical Center (US) 2001-03-28 EP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
WO-2000001410-A9 METHODS OF INHIBITING PROLIFERATIVE DISEASES BY INHIBITING TGF-BETA MEDIATED ANGIOGENESIS BETH ISRAEL HOSPITAL (US) 2000-05-25 WO claimed
WO-2000001410-A1 METHODS OF INHIBITING PROLIFERATIVE DISEASES BY INHIBITING TGF-BETA MEDIATED ANGIOGENESIS BETH ISRAEL DEACONESS MEDICAL CENTER (US) 2000-01-13 WO claimed
WO-1999065940-A1 ANTI-ANGIOGENIC PROTEINS AND METHODS OF USE THEREOF BETH ISRAEL DEACONESS MEDICAL CENTER (US) 1999-12-23 WO claimed
US-5811547-A Method for inducing crystalline state transition in medicinal substance NIPPON SHINYAJU CO., LTD. (JP) 1998-09-22 US claimed
EP-0753301-A1 Combination of benzimidazoles having angiotensin-II antagonistic activity with diuretics TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-15 EP claimed
EP-0628313-A1 Combination of benzimidazoles having angiotensin-II antagonistic activity with dinretics or calcium antagonists TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-14 EP claimed