Etomoxir

Etomoxir

SCHEMBL49075

CCOC(=O)[C@@]1(CCCCCCOc2ccc(Cl)cc2)CO1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 1.00
LMNA P02545 1/20 1.00
MAPT P10636 1/20 1.00
MAPK1 P28482 1/20 1.00
CPT1A P50416 1/20 0.51
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
HRH3 Q9Y5N1 9/20 0.42
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rac-Etomoxir SCHEMBL15256787 1.00 ABCB11 (1.00) ABCB11LMNAMAPTMAPK1CPT1A
SCHEMBL954683 1.00 ABCB11 (1.00) ABCB11LMNAMAPTMAPK1CPT1A
Rac-Etomoxir SCHEMBL681359 1.00 ABCB11 (1.00) ABCB11LMNAMAPTMAPK1CPT1A
Etomoxir SCHEMBL12813827 0.99 MAPT (0.98) ABCB11LMNAMAPTMAPK1CPT1A
Etomoxir SCHEMBL5883664 0.99 MAPT (0.98) ABCB11LMNAMAPTMAPK1CPT1A
Rac-Etomoxir SCHEMBL2141141 0.98 MAPT (0.95) ABCB11LMNAMAPTMAPK1CPT1A
Etomoxir SCHEMBL22206060 0.93 MAPT (0.87) ABCB11LMNAMAPTMAPK1CPT1A
SCHEMBL11294309 0.90 LMNA (0.82) ABCB11LMNAMAPTMAPK1CPT1A
SCHEMBL14769764 0.90 MAPT (0.82) ABCB11LMNAMAPTMAPK1CPT1A
SCHEMBL11288224 0.89 MAPT (0.80) ABCB11LMNAMAPTMAPK1HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3811 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260076954-A1 COMPOSITIONS AND METHODS FOR REDUCING CANCER STEM CELLS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2026-03-19 US claimed
US-12544368-B2 Compositions and methods for reducing cancer stem cells THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2026-02-10 US claimed
EP-4678750-A1 REPLICON DNA, CLONING VECTOR, SCREENING KIT, SCREENING METHOD, ANTI-NOBECOVIRUS AGENT, BETA-CORONAVIRUS PROLIFERATION INHIBITOR, PAN BETA-CORONAVIRUS INHIBITOR, VIRUS PROLIFERATION INHIBITOR, HEPATITIS C VIRUS PROLIFERATION INHIBITOR, AND METHOD FOR SCREENING THERAPEUTIC AGENT FOR VIRAL INFECTIOUS DISEASE Kagoshima University (JP) 2026-01-14 EP claimed
US-20250297321-A1 METHOD FOR DETECTING METABOLIC REPROGRAMING OF CANCER TOWARDS FATTY ACIDS METABOLISM INST NAT SANTE RECH MED (FR) 2025-09-25 US claimed
EP-3976197-B1 THERAPEUTICS AND METHODS FOR PREDICTING AND OVERCOMING ENDOCRINE RESISTANCE IN BREAST CANCER LUNELLA BIOTECH INC (CA) 2025-07-16 EP claimed
EP-3956663-B1 A METHOD OF PROFILING THE ENERGETIC METABOLISM OF A POPULATION OF CELLS INST NAT SANTE RECH MED (FR) 2025-02-12 EP claimed
US-20250011719-A1 NEW METHOD FOR IMPROVING QUALITY OF PLATELETS SHANGHAI SYNVIDA BIOTECHNOLOGY CO. LTD. (CN) 2025-01-09 US claimed
EP-4469602-A1 METHOD FOR DETECTING METABOLIC REPROGRAMING OF CANCER TOWARDS FATTY ACIDS METABOLISM Université Paris Cité (FR) 2024-12-04 EP claimed
CN-119055773-A Drug for reversing drug resistance of EGFR-TKI of third generation lung cancer 华中农业大学 2024-12-03 CN claimed
WO-2024214687-A1 REPLICON DNA, CLONING VECTOR, SCREENING KIT, SCREENING METHOD, ANTI-NOBECOVIRUS AGENT, BETA-CORONAVIRUS PROLIFERATION INHIBITOR, PAN BETA-CORONAVIRUS INHIBITOR, VIRUS PROLIFERATION INHIBITOR, HEPATITIS C VIRUS PROLIFERATION INHIBITOR, AND METHOD FOR SCREENING THERAPEUTIC AGENT FOR VIRAL INFECTIOUS DISEASE 国立大学法人 鹿児島大学 2024-10-17 WO claimed
EP-1226830-A2 Combination therapy involving a sodium-hydrogen exchanger type 1 or NHE-1 inhibitor for use in treatment of ischemia Pfizer Products Inc. (US) 2002-07-31 EP claimed
US-20020099075-A1 COMBINATION THERAPY TRACEY WAYNE R (US) 2002-07-25 US claimed
US-6423705-B1 FOR ISCHEMIA BY ADMINISTERING AN NHE-1 INHIBITOR AND A SECOND COMPOUND SELECTED FROM COMPLEMENT MODULATOR, METABOLIC MODULATOR, ANTIAPOPTOTIC AGENT, NITRIC OXIDE SYNTHASE-RELATED AGENT, AND AN ENZYME/PROTEIN MODULATOR PFIZER INC. 2002-07-23 US claimed
WO-2002056022-A2 DIAGNOSTICS, DRUG SCREENING AND TREATMENT FOR CANCER MINERVA BIOTECHNOLOGIES CORP (US) 2002-07-18 WO claimed
US-6399601-B1 ANTIDIABETIC AGENTS; NERVOUS SYSTEM DISORDERS; ANTICHOLESTEROL AGENTS PFIZER INC. 2002-06-04 US claimed
US-20020013268-A1 Synergistic effect of a sulfonylurea and/or non-sulfonylurea Kchannel blocker, and a phosphodiesterase 3 type inhibitor FRYBURG DAVID A (US) 2002-01-31 US claimed
EP-1145717-A2 Synergistic effect of a sulfonylurea and/or non-sulfonylurea K plus ATP channel blocker, and a phosphodiesterase 3 type inhibitor Pfizer Products Inc. (US) 2001-10-17 EP claimed
EP-1136071-A2 Use of glycogen phosphorylase inhibitors Pfizer Products Inc. (US) 2001-09-26 EP claimed
WO-2001034145-A1 TREATING CANCER BY INCREASING INTRACELLULAR MALONYL COA LEVELS THE JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (US) 2001-05-17 WO claimed
EP-1088824-A2 Bicyclic pyrrolyl amides as glycogen phosphorylase inhibitors Pfizer Products Inc. (US) 2001-04-04 EP claimed