Rac-Etomoxir

Rac-Etomoxir

SCHEMBL681359

CCOC(=O)C1(CCCCCCOc2ccc(Cl)cc2)CO1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 1.00
LMNA P02545 1/20 1.00
MAPT P10636 1/20 1.00
MAPK1 P28482 1/20 1.00
CPT1A P50416 1/20 0.51
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
HRH3 Q9Y5N1 9/20 0.42
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rac-Etomoxir SCHEMBL15256787 1.00 ABCB11 (1.00) ABCB11LMNAMAPTMAPK1CPT1A
SCHEMBL954683 1.00 ABCB11 (1.00) ABCB11LMNAMAPTMAPK1CPT1A
Etomoxir SCHEMBL49075 1.00 ABCB11 (1.00) ABCB11LMNAMAPTMAPK1CPT1A
Etomoxir SCHEMBL12813827 0.99 MAPT (0.98) ABCB11LMNAMAPTMAPK1CPT1A
Etomoxir SCHEMBL5883664 0.99 MAPT (0.98) ABCB11LMNAMAPTMAPK1CPT1A
Rac-Etomoxir SCHEMBL2141141 0.98 MAPT (0.95) ABCB11LMNAMAPTMAPK1CPT1A
Etomoxir SCHEMBL22206060 0.93 MAPT (0.87) ABCB11LMNAMAPTMAPK1CPT1A
SCHEMBL11294309 0.90 LMNA (0.82) ABCB11LMNAMAPTMAPK1CPT1A
SCHEMBL14769764 0.90 MAPT (0.82) ABCB11LMNAMAPTMAPK1CPT1A
SCHEMBL11288224 0.89 MAPT (0.80) ABCB11LMNAMAPTMAPK1HRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 137 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200330400-A1 METHODS FOR THE TREATMENT OF CANCER USING COENZYME Q10 AND FATTY ACID METABOLISM INHIBITORS BERG LLC 2020-10-22 US claimed
EP-2310003-B1 INHIBITORS OF CARNITIN-PALMITOYL-TRANSFERASE-1 FOR THE TREATMENT AND PREVENTION OF DISORDERS CAUSED BY DELIPIDATION OF NEURAL TISSUE META IQ APS (DK) 2020-02-12 EP claimed
WO-2017161205-A1 METHODS FOR THE TREATMENT OF CANCER USING COENZYME Q10 AND FATTY ACID METABOLISM INHIBITORS BERG LLC (US) 2017-09-21 WO claimed
EP-2445506-B1 THE USE OF SPINOSYNS AND SPINOSYN COMPOSITIONS AGAINST DISEASES CAUSED BY PROTOZOANS, VIRAL INFECTIONS AND CANCER ENTARCO SA (GR) 2014-12-31 EP claimed
US-8741949-B2 Inhibitors of carnitin-palmitoyl-tranferase-1 for the treatment and prevention of disorders caused by delipidation of neural tissue META-IQ APS (DK) 2014-06-03 US claimed
WO-2014018801-A1 DIAGNOSIS AND TREATMENT OF CANCER USING DIFFERENTIALLY EXPRESSED STARVATION MARKERS THE TEXAS A&M UNIVERSITY SYSTEM (US) 2014-01-30 WO claimed
WO-2013071029-A1 METHODS AND PRODUCTS FOR GENERATING OILS THE TEXAS A&M UNIVERSITY SYSTEM (US) 2013-05-16 WO claimed
US-20130056683-A1 COMPOSITIONS AND METHODS FOR PROMOTING FATTY ACID PRODUCTION IN PLANTS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2013-03-07 US claimed
WO-2012135632-A2 METHODS OF TREATING A SUBJECT HAVING BEEN EXPOSED TO A CATASTROPHIC EVENT THE TEXAS A&M UNIVERSITY SYSTEM (US) 2012-10-04 WO claimed
EP-2486140-A2 COMPOSITIONS AND METHODS FOR PROMOTING FATTY ACID PRODUCTION IN PLANTS Regents of the University of Colorado (US) 2012-08-15 EP claimed
EP-1275390-B1 Medicament for treatment of heart failure WOLF HORST P O (DE) 2005-11-02 EP claimed
EP-1549398-A1 INHIBITORS OF THE FATTY ACID OXIDATION FOR THE PROPHYLAXIS AND/OR THE TREATMENT OF CHRONIC AND/OR ATOPIC SKIN DISEASES MediGene Aktiengesellschaft (DE) 2005-07-06 EP claimed
US-20050004173-A1 Inhibitors of fatty acid oxidation for prophylaxis and treatment of diseases related to mitochondrial dysfunction MEDIGENE AG (DE) 2005-01-06 US claimed
WO-2004026405-A1 INHIBITORS OF THE FATTY ACID OXIDATION FOR THE PROPHYLAXIS AND/OR THE TREATMENT OF CHRONIC AND/OR ATOPIC SKIN DISEASES MEDIGENE AKTIENGESELLSCHAFT (DE) 2004-04-01 WO claimed
WO-2003037323-A2 INHIBITORS OF THE FATTY ACID OXIDATION FOR PROPHYLAXIS AND TREATMENT OF DISEASES RELATED TO MITOCHONDRIAL DYSFUNCTION MEDIGENE AG Gesellschaft für Molekularbiologische Kardiologie und Onkologie (DE) 2003-05-08 WO claimed
US-5739159-A Medicaments for the treatment of cardiac insufficiency WOLF HORST (DE) 1998-04-14 US claimed
EP-0231367-B1 USE OF OXIRANCARBOXYLIC ACIDS FOR THE TREATMENT OF HYPERLIPEMIA Wolf, Horst P.O., Dr. (DE) 1991-07-24 EP claimed
US-4933365-A ANTIFLAMMATORY AGENTS, ANTIALLERGENS AMERICAN HOME PRODUCTS CORPORATION (US) 1990-06-12 US claimed
WO-1989005142-A1 PHOSPHOLIPASE A2 INHIBITORS AMERICAN HOME PRODUCTS CORPORATION (US) 1989-06-15 WO claimed
EP-0046590-B1 PHEN(ALK)OXY-SUBSTITUTED OXIRANE-CARBOXYLIC ACIDS, PROCESS FOR THEIR PREPARATION, THEIR USE AND DRUGS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1985-05-22 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004173-A1 Inhibitors of fatty acid oxidation for prophylaxis and treatment of diseases related to mitochondrial dysfunction CPT1A, CPT2, CPT1B ABCB11 2356/4885LMNA 2830/4885MAPT 1990/4885
US-20200330400-A1 METHODS FOR THE TREATMENT OF CANCER USING COENZYME Q10 AND FATTY ACID METABOLISM INHIBITORS CPT1B, CPT2, CPT1A ABCB11 1461/4885LMNA 1667/4885MAPT 2554/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.