SCHEMBL490938

SCHEMBL490938

O=C(O)C(Cc1ccccc1O)C(=O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.60
AKR1B1 P15121 1/20 0.59
HSPA5 P11021 1/20 0.50
HIF1A Q16665 2/20 0.45
CYP2D6 P10635 1/20 0.45
TSHR P16473 1/20 0.45
TAAR1 Q96RJ0 1/20 0.43
CYP1A2 P05177 1/20 0.43
CTNNB1 P35222 1/20 0.43
SLC7A5 Q01650 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CYP2C19 P33261 1/20 0.42
POLB P06746 1/20 0.42
MAPK1 P28482 1/20 0.42
CA12 O43570 2/20 0.42
CA2 P00918 2/20 0.42
IDO1 P14902 1/20 0.42
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10457141 0.88 AKR1B1 (0.52) KMT2AAKR1B1HSPA5HIF1ACYP2D6
SCHEMBL7388453 0.85 AKR1B1 (0.57) KMT2AAKR1B1HSPA5HIF1ACYP2D6
SCHEMBL7590369 0.84 AKR1B1 (0.47) KMT2AAKR1B1HSPA5TAAR1PKM
SCHEMBL6695633 0.83 AKR1B1 (0.50) KMT2AAKR1B1HSPA5HIF1ACYP2D6
SCHEMBL8319229 0.83 SMN1; SMN2 (0.56) KMT2AAKR1B1HSPA5HIF1ACYP2D6
SCHEMBL16815384 0.83 SMN1; SMN2 (0.56) KMT2AAKR1B1HSPA5HIF1ACYP2D6
SCHEMBL490685 0.83 KMT2A (0.52) KMT2AAKR1B1CTNNB1CYP2C19CA12
SCHEMBL18341946 0.83 SMN1; SMN2 (0.56) KMT2AAKR1B1HSPA5HIF1ACYP2D6
SCHEMBL29367333 0.83 SMN1; SMN2 (0.56) KMT2AAKR1B1HSPA5HIF1ACYP2D6
SCHEMBL352381 0.83 SMN1; SMN2 (0.56) KMT2AAKR1B1HSPA5HIF1ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8268293-B2 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives MERCK PATENT GMBH (DE) 2012-09-18 US disclosed
US-8106233-B2 Applying di-2-ethylhexyl 4-hydroxy-3,5-dimethoxy-benzylmalonate; protective action against UV rays, oxidative stress on body cells, counters skin ageing MERCK PATENT GMBH (DE) 2012-01-31 US disclosed
US-20080171004-A1 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives MERCK PATENT GMBH (DE) 2008-07-17 US disclosed
US-20080152603-A1 Antioxidants SUSONITY Commercial GmbH (DE) 2008-06-26 US disclosed
EP-1871735-A1 ANTIOXIDANTS Merck Patent GmbH (DE) 2008-01-02 EP disclosed
EP-1871339-A1 UV PROTECTION Merck Patent GmbH (DE) 2008-01-02 EP disclosed
WO-2006111233-A1 ANTIOXIDANTS MERCK PATENT GMBH (DE) 2006-10-26 WO disclosed
WO-2006111234-A1 UV PROTECTION MERCK PATENT GMBH (DE) 2006-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080152603-A1 Antioxidants GPX4, GPX1, CAT KMT2A 4023/4885AKR1B1 244/4885HSPA5 1029/4885
US-20080171004-A1 Using compounds which do not themselves exhibit significant UV absorption in the UV-A or UV-B region, but are reactive under use conditions, such as 4-hydroxyphenylpropionic acid, or 2-ethylhexyl 4-hydroxy-3,5-dimethoxycinnamate, or polysiloxanes which contain benzylidenemalonic acid derivatives HPD, HAAO, UGT1A6 KMT2A 1522/4885AKR1B1 1345/4885HSPA5 681/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.