SCHEMBL4912940

SCHEMBL4912940

O=C(COc1ccc(Cl)c(F)c1)Nc1ccc(O)cc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.58
KDM4E B2RXH2 2/20 0.54
ALDH1A1 P00352 1/20 0.54
HSD17B10 Q99714 1/20 0.54
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.52
CASP3 P42574 1/20 0.51
SENP8 Q96LD8 1/20 0.51
SENP7 Q9BQF6 1/20 0.51
SENP6 Q9GZR1 1/20 0.51
MAPT P10636 1/20 0.50
ATF4 P18848 4/20 0.48
DVL1 O14640 1/20 0.48
SERPINE1 P05121 1/20 0.48
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.45
POLB P06746 1/20 0.45
G6PD P11413 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4905601 0.91 HCAR2 (0.58) HCAR2KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL4913841 0.87 KMT2A (0.68) HCAR2KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL4912174 0.84 HCAR2 (0.58) HCAR2KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL3556752 0.83 ATF4 (0.47) HCAR2KMT2AMEN1CASP3SENP8
SCHEMBL4904904 0.82 ALDH1A1 (0.59) HCAR2KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL4914768 0.82 KDM4E (0.59) HCAR2KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL4904826 0.81 KDM4E (0.63) HCAR2KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL4914734 0.81 SERPINE1 (0.62) HCAR2KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL22189806 0.81 KDM4C (0.51) HCAR2KMT2AMEN1CASP3SENP8
SCHEMBL4905629 0.80 ALDH1A1 (0.65) HCAR2KDM4EALDH1A1HSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2008-10-30 US claimed
US-7408078-B2 Anthranilic acid derivatives useful in treating infection with hepatitis C virus WYETH (US) 2008-08-05 US claimed
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus VIROPHARMA INCORPORATED 2005-01-06 US claimed
WO-2004091724-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2004-10-28 WO claimed
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2008-10-30 US disclosed
US-7408078-B2 Anthranilic acid derivatives useful in treating infection with hepatitis C virus WYETH (US) 2008-08-05 US disclosed
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus VIROPHARMA INCORPORATED 2005-01-06 US disclosed
WO-2004091724-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2004-10-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus HCCS, ALAD, HAVCR2 HCAR2 103/4885KDM4E 2214/4885ALDH1A1 271/4885
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS HCCS, ALAD, HAVCR2 HCAR2 103/4885KDM4E 2214/4885ALDH1A1 271/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.