Allopurinol

Allopurinol

SCHEMBL4916844

Nc1ncnc2n[nH]cc12.Oc1ncnc2[nH]ncc12

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

XDH

The experimentally established mechanism targets of Allopurinol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH known ✓ P47989 1/20 0.57
RET P07949 1/20 0.57
PI4KA P42356 1/20 0.57
LRRK2 Q5S007 1/20 0.57
PI4K2B Q8TCG2 1/20 0.57
PI4K2A Q9BTU6 1/20 0.57
PI4KB Q9UBF8 1/20 0.57
CYP1A2 P05177 2/20 0.39
PDPK1 O15530 2/20 0.39
CHEK1 O14757 1/20 0.38
AURKA O14965 1/20 0.38
TTBK1 Q5TCY1 1/20 0.36
LMNA P02545 1/20 0.35
MAPK1 P28482 2/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGDS O60760 1/20 0.35
AKT2 P31751 2/20 0.34
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
CCNA1 P78396 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Allopurinol SCHEMBL29693720 0.80 XDH (0.61) RETPI4KAXDHLRRK2PI4K2B
Allopurinol SCHEMBL4627 0.80 XDH (0.61) RETPI4KAXDHLRRK2PI4K2B
SCHEMBL11362 0.80 PI4KA (0.45) RETPI4KAXDHLRRK2PI4K2B
Allopurinol SCHEMBL4708652 0.80 XDH (0.61) RETPI4KAXDHLRRK2PI4K2B
Allopurinol SCHEMBL21362860 0.78 XDH (0.59) RETPI4KAXDHLRRK2PI4K2B
Allopurinol SCHEMBL137084 0.78 XDH (0.59) RETPI4KAXDHLRRK2PI4K2B
Allopurinol SCHEMBL7202468 0.78 XDH (0.59) RETPI4KAXDHLRRK2PI4K2B
Hydrochloric Acid SCHEMBL1741651 0.78 PI4KA (0.44) RETPI4KAXDHLRRK2PI4K2B
Hydrochloric Acid SCHEMBL14742344 0.78 PI4KA (0.44) RETPI4KAXDHLRRK2PI4K2B
Allopurinol SCHEMBL27973688 0.78 XDH (0.59) RETPI4KAXDHLRRK2PI4K2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080089957-A1 Monocotyledon plant indications extract compositions, method of preparation and pharmaceutical compositions containing them ACADEMIA SINICA (TW) 2008-04-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080089957-A1 Monocotyledon plant indications extract compositions, method of preparation and pharmaceutical compositions containing them OAT, TPMT, NUDT1 XDH 5/4885RET 3750/4885PI4KA 4187/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.