SCHEMBL4921708

SCHEMBL4921708

OC(c1nc2ccccc2[nH]1)C(O)c1nc2ccccc2[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 1.00
GAA P10253 2/20 0.73
L3MBTL1 Q9Y468 2/20 0.68
ALOX12 P18054 1/20 0.68
ALDH1A1 P00352 4/20 0.66
POLB P06746 2/20 0.66
MLKL Q8NB16 3/20 0.60
USP2 O75604 2/20 0.58
ALPL P05186 1/20 0.58
ALPI P09923 1/20 0.58
ALPG P10696 1/20 0.58
HPGD P15428 1/20 0.58
HTT P42858 1/20 0.58
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
KDM4E B2RXH2 1/20 0.54
ABCB11 O95342 1/20 0.54
TP53 P04637 1/20 0.54
PKM P14618 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19425618 0.92 IDO1 (0.85) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL19425511 0.92 IDO1 (0.85) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL15221577 0.89 IDO1 (0.79) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL16376072 0.89 IDO1 (0.79) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL7101160 0.89 IDO1 (0.79) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL7946544 0.88 IDO1 (0.78) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL12858901 0.84 IDO1 (0.72) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL15294554 0.84 ALOX12 (0.73) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL2674618 0.84 IDO1 (0.72) IDO1GAAL3MBTL1ALOX12ALDH1A1
SCHEMBL2673705 0.84 IDO1 (0.72) IDO1GAAL3MBTL1ALOX12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104829634-B A kind of thirty-two nucleus copper complex and preparation method thereof 山西大学 2016-09-28 CN claimed
EP-3318561-B1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC (US) 2021-12-22 EP disclosed
CN-104829634-B A kind of thirty-two nucleus copper complex and preparation method thereof 山西大学 2016-09-28 CN disclosed
CN-104829634-A Tridodenuclear copper complex and preparation method thereof UNIV SHANXI 2015-08-12 CN disclosed
US-20080280933-A1 BENZIMIDAZOLYL COMPOUNDS EFREMOV IVAN 2008-11-13 US disclosed
US-20050020654-A1 Novel PPAR agonists, pharmaceutical compositions and uses thereof BETHESDA PHARMACEUTICALS, INC. 2005-01-27 US disclosed
WO-2004082621-A2 NOVEL PPAR AGONISTS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BETHESDA PHARMACEUTICALS, INC. (US) 2004-09-30 WO disclosed
EP-0276942-B1 6-BETA(SUBSTITUTED)-(S)-HYDROXYMETHYLPENICILLANIC ACIDS AND DERIVATIVES THEREOF PFIZER INC. (US) 1992-04-01 EP disclosed
US-4782050-A BACTERICIDES PFIZER INC. (US) 1988-11-01 US disclosed
EP-0276942-A1 6-Beta(substituted)-(S)-hydroxymethylpenicillanic acids and derivatives thereof PFIZER INC. (US) 1988-08-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050020654-A1 Novel PPAR agonists, pharmaceutical compositions and uses thereof PPARG, PPARD, PPARA IDO1 1134/4885GAA 1820/4885L3MBTL1 4796/4885
US-20080280933-A1 BENZIMIDAZOLYL COMPOUNDS PAICS, TMBIM6, ABCG2 IDO1 2062/4885GAA 44/4885L3MBTL1 4582/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.