SCHEMBL4922985

SCHEMBL4922985

CN(C(=O)OCc1cc(-c2ccccc2)n(S(=O)(=O)c2cccnc2Cl)c1)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.38
POLB P06746 1/20 0.37
SLC16A3 O15427 10/20 0.36
ACLY P53396 1/20 0.36
SLC16A1 P53985 6/20 0.34
MCTS1 Q9ULC4 5/20 0.34
KAT8 Q9H7Z6 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CNR2 P34972 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1156675 0.82 HTR2C (0.41) POLBSLC16A3ACLYSLC16A1MCTS1
SCHEMBL1156338 0.81 ACLY (0.39) SLC16A3ACLYMEN1KMT2ACNR2
SCHEMBL1156677 0.78 ACLY (0.37) RXFP1POLBSLC16A3ACLYSLC16A1
SCHEMBL1580757 0.77 ACLY (0.39) SLC16A3ACLYKAT8MEN1KMT2A
Hydrochloric Acid SCHEMBL1156903 0.76 ACLY (0.39) SLC16A3ACLYKAT8MEN1KMT2A
SCHEMBL1156674 0.76 ACLY (0.38) SLC16A3ACLYKAT8PTGDR2
SCHEMBL1156341 0.76 ACLY (0.41) ACLYMEN1KMT2APTGDR2
SCHEMBL4566726 0.72 CTSD (0.31) RXFP1
SCHEMBL1156292 0.71 ACLY (0.40) ACLYMEN1KMT2ACHRM1
SCHEMBL4566702 0.70 ALDH1A1 (0.35) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed