SCHEMBL492454

SCHEMBL492454

FC(F)(F)OC1CCNC1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 9/20 0.35
HTR1A P08908 6/20 0.35
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 3/20 0.33
KCNH2 Q12809 3/20 0.33
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
PRKCZ Q05513 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23299878 1.00 SLC6A2 (0.35) SLC6A2HTR1ACHRNB2CHRNA4SLC6A4
SCHEMBL22488570 1.00 SLC6A2 (0.35) SLC6A2HTR1ACHRNB2CHRNA4SLC6A4
Hydrochloric Acid SCHEMBL29159595 0.98 SLC6A2 (0.34) SLC6A2HTR1ACHRNB2CHRNA4SLC6A4
Hydrochloric Acid SCHEMBL22468398 0.98 SLC6A2 (0.34) SLC6A2HTR1ACHRNB2CHRNA4SLC6A4
Hydrochloric Acid SCHEMBL25313788 0.98 SLC6A2 (0.34) SLC6A2HTR1ACHRNB2CHRNA4SLC6A4
SCHEMBL29159638 0.86 CHRNB2 (0.37) SLC6A2HTR1ACHRNB2CHRNA4CHRM2
SCHEMBL28086801 0.86 CHRNB2 (0.37) SLC6A2HTR1ACHRNB2CHRNA4CHRM2
SCHEMBL15740845 0.85 HRH1 (0.35) SLC6A2HTR1ASLC6A3
Hydrochloric Acid SCHEMBL29159632 0.85 CHRNB2 (0.36) SLC6A2HTR1ACHRNB2CHRNA4CHRM2
Hydrochloric Acid SCHEMBL15740523 0.83 HTR2C (0.35) SLC6A2HTR1ASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025264645-A1 SODIUM CHANNEL BLOCKING COMPOUNDS, DERIVATIVES THEREOF, AND METHODS OF THEIR USE LATIGO BIOTHERAPEUTICS, INC. (US) 2025-12-26 WO disclosed
WO-2025092827-A1 EPOXY COMPOUND AND USE THEREOF 上海汇伦医药股份有限公司 2025-05-08 WO disclosed
US-20250145594-A1 MODULATORS OF THE INTEGRATED STRESS PATHWAY ABBVIE INC. 2025-05-08 US disclosed
CN-115925698-B Imidazo [4,5-g ] quinolin-2-one compounds and their use as pesticides 中新科农(山东)生态农业有限公司 2025-02-25 CN disclosed
US-20240207263-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF SUZHOU ZANRONG PHARMA LIMITED (CN) 2024-06-27 US disclosed
CN-117580824-A Modulators of integrated stress pathways 卡里科生命科学有限责任公司 2024-02-20 CN disclosed
US-20230374036-A1 KRAS G12D MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-11-23 US disclosed
US-20230339981-A1 KRAS G12D MODULATING COMPOUNDS GILEAD SCIENCES, INC. 2023-10-26 US disclosed
WO-2023205719-A1 KRAS G12D MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2023-10-26 WO disclosed
CN-114891003-B Novel dihydropyrimidine compound, intermediate or salt, and preparation method and application thereof 成都施贝康生物医药科技有限公司 2023-10-13 CN disclosed
WO-2022094244-A1 MODULATORS OF THE INTEGRATED STRESS PATHWAY CALICO LIFE SCIENCES LLC (US) 2022-05-05 WO disclosed
WO-2020198058-A1 INHIBITORS OF RAF KINASES KINNATE BIOPHARMA INC. (US) 2020-10-01 WO disclosed
CN-108129472-A A kind of (trifluoromethoxy) pyrrolidines benzamide compound and its purposes in thrombopenia is treated 窦玉玲 2018-06-08 CN disclosed
US-8273891-B2 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof MEMORY PHARMACEUTICALS CORPORATION (US) 2012-09-25 US disclosed
US-8106066-B2 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof MEMORY PHARMACEUTICALS CORPORATION (US) 2012-01-31 US disclosed
US-20100137288-A1 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, PYRAZOLOPYRIDINES, ISOTHIAZOLOPYRIDINES, AND PREPARATION AND USES THEREOF SCHUMACHER RICHARD 2010-06-03 US disclosed
CN-101312968-A Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof MEMORY PHARM CORP (US) 2008-11-26 CN disclosed
EP-1940833-A1 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, PYRAZOLOPYRIDINES, ISOTHIAZOLOPYRIDINES, AND PREPARATION AND USES THEREOF Memory Pharmaceuticals Corporation (US) 2008-07-09 EP disclosed
US-20070078147-A1 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof MEMORY PHARMACEUTICALS CORPORATION 2007-04-05 US disclosed
WO-2007038367-A1 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, PYRAZOLOPYRIDINES, ISOTHIAZOLOPYRIDINES, AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2007-04-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100137288-A1 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, PYRAZOLOPYRIDINES, ISOTHIAZOLOPYRIDINES, AND PREPARATION AND USES THEREOF CHRNA7, CHRNA5, CHRNA2 SLC6A2 864/4885HTR1A 626/4885CHRNB2 10/4885
US-20250145594-A1 MODULATORS OF THE INTEGRATED STRESS PATHWAY ATF4, ATF1, DDIT3 SLC6A2 1180/4885HTR1A 1457/4885CHRNB2 2826/4885
US-20230339981-A1 KRAS G12D MODULATING COMPOUNDS KRAS, NRAS, HRAS SLC6A2 4859/4885HTR1A 4791/4885CHRNB2 4815/4885
US-20230374036-A1 KRAS G12D MODULATING COMPOUNDS KRAS, NRAS, HRAS SLC6A2 4859/4885HTR1A 4791/4885CHRNB2 4815/4885
US-20240207263-A1 SELECTIVE MODULATORS OF ATAXIA TELANGIECTASIA MUTATED (ATM) KINASE AND USES THEREOF ATM, CHEK2, CHEK1 SLC6A2 4804/4885HTR1A 4619/4885CHRNB2 2441/4885
US-20070078147-A1 Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof CHRNA7, CHRNA5, CHRNA2 SLC6A2 864/4885HTR1A 626/4885CHRNB2 10/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.