SCHEMBL4928762

SCHEMBL4928762

CCc1oc(-c2ccc(C)cc2)nc1COCCl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.43
PPARA Q07869 4/20 0.43
TARBP2 Q15633 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.38
POLB P06746 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 4/20 0.37
ALDH1A1 P00352 3/20 0.37
TP53 P04637 3/20 0.37
RAB9A P51151 3/20 0.37
HPGD P15428 2/20 0.37
NPC1 O15118 2/20 0.37
HSD17B10 Q99714 2/20 0.37
LMNA P02545 2/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
PPARD Q03181 1/20 0.36
KMT2A Q03164 3/20 0.35
ALOX12 P18054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1929665 0.84 PPARG (0.47) PPARGPPARATARBP2SMN1; SMN2POLB
SCHEMBL4928637 0.82 CYP1A2 (0.41) PPARGPPARASMN1; SMN2POLBMAPT
SCHEMBL1048319 0.78 PPARG (0.47) PPARGPPARATARBP2SMN1; SMN2POLB
SCHEMBL5855879 0.78 PPARG (0.56) PPARGPPARATARBP2SMN1; SMN2POLB
SCHEMBL5182375 0.78 PPARA (0.43) PPARGPPARAMAPTKDM4EALDH1A1
SCHEMBL4921322 0.77 VDR (0.47) PPARGPPARASMN1; SMN2MAPTKDM4E
SCHEMBL18095687 0.75 PPARG (0.54) PPARGPPARATARBP2SMN1; SMN2POLB
SCHEMBL4925797 0.75 KMT2A (0.40) SMN1; SMN2POLBMAPTKDM4EALDH1A1
SCHEMBL4929598 0.72 KDM4E (0.56) PPARGPPARATARBP2KDM4ERAB9A
SCHEMBL1930635 0.72 HSD17B10 (0.43) TARBP2SMN1; SMN2POLBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080015238-A1 CYCLOALKYLMETHOXY-SUBSTITUTED ACETIC ACID DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-01-17 US disclosed
US-7259177-B2 Cycloalkylmethoxy-substituted acetic acid derivatives, processes for their preparation and their use as pharmaceuticals SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2007-08-21 US disclosed
US-20050101637-A1 Cycloalkylmethoxy-substituted acetic acid derivatives, processes for their preparation and their use as pharmaceuticals AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2005-05-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080015238-A1 CYCLOALKYLMETHOXY-SUBSTITUTED ACETIC ACID DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS GPR119, PC, ACADM PPARG 80/4885PPARA 122/4885TARBP2 4538/4885
US-20050101637-A1 Cycloalkylmethoxy-substituted acetic acid derivatives, processes for their preparation and their use as pharmaceuticals GPR119, PC, CPT1A PPARG 99/4885PPARA 132/4885TARBP2 4532/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.