SCHEMBL4930331

SCHEMBL4930331

N#Cc1ccc(Cn2cc(CC(N)C(=O)NO)c3ccccc32)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.59
HTT P42858 2/20 0.59
CYP19A1 P11511 3/20 0.54
POLB P06746 1/20 0.52
MAPT P10636 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
HDAC6 Q9UBN7 9/20 0.49
HDAC1 Q13547 7/20 0.49
HDAC10 Q969S8 5/20 0.49
HDAC8 Q9BY41 5/20 0.49
KMT2A Q03164 1/20 0.49
HDAC2 Q92769 4/20 0.47
HDAC3 O15379 2/20 0.47
NCOR2 Q9Y618 2/20 0.47
PTGS2 P35354 1/20 0.47
NPM1 P06748 1/20 0.45
HDAC9 Q9UKV0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4930338 1.00 LMNA (0.59) LMNAHTTCYP19A1POLBMAPT
SCHEMBL4933909 0.83 HDAC6 (0.53) HDAC6HDAC1HDAC10HDAC8KMT2A
SCHEMBL4927847 0.83 HTR6 (0.54) MAPTHDAC6HDAC1HDAC10HDAC8
SCHEMBL4933914 0.83 HDAC6 (0.53) HDAC6HDAC1HDAC10HDAC8KMT2A
SCHEMBL4927838 0.83 HTR6 (0.54) MAPTHDAC6HDAC1HDAC10HDAC8
SCHEMBL4926554 0.81 HDAC6 (0.47) LMNAHTTMAPTHDAC6HDAC1
SCHEMBL4926564 0.81 HDAC6 (0.47) LMNAHTTMAPTHDAC6HDAC1
SCHEMBL4935914 0.81 HDAC6 (0.47) LMNAHTTMAPTHDAC6HDAC1
SCHEMBL4932173 0.81 ALDH1A1 (0.51) LMNACYP19A1POLBMAPTKMT2A
SCHEMBL4930609 0.81 ALDH1A1 (0.51) LMNACYP19A1POLBMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080132539-A1 Hydroxamic Acid Derivative And Age Generation Inhibitor Containing The Derivative KUREHA CORPORATION (JP) 2008-06-05 US disclosed
EP-1707560-A1 HYDROXAMIC ACID DERIVATIVE AND AGE GENERATION INHIBITOR CONTAINING THE DERIVATIVE Kureha Corporation (JP) 2006-10-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080132539-A1 Hydroxamic Acid Derivative And Age Generation Inhibitor Containing The Derivative HDAC5, HDAC1, HDAC9 LMNA 1237/4885HTT 1087/4885CYP19A1 792/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.