SCHEMBL4933162

SCHEMBL4933162

O=C(O)CNC(=O)c1cc(Cl)c(OCc2cc(NC3CCC3)cc(C(F)(F)F)c2)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 12/20 0.42
RHOC P08134 3/20 0.37
RHOA P61586 3/20 0.37
CCR2 P41597 3/20 0.35
USP5 P45974 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5717942 0.96 MRGPRX4 (0.39) MRGPRX4RHOCRHOACCR2USP5
SCHEMBL4929949 0.91 THRA (0.41) MRGPRX4RHOCRHOACCR2USP5
SCHEMBL5717949 0.89 MRGPRX4 (0.39) MRGPRX4RHOCRHOACCR2
SCHEMBL4931877 0.88 PDE4A (0.35) MRGPRX4USP5
SCHEMBL4926882 0.88 PDE4A (0.36) MRGPRX4USP5
SCHEMBL4931806 0.86 F2 (0.39) USP5
SCHEMBL4932229 0.85 PPARD (0.43) MRGPRX4RHOCRHOA
SCHEMBL4922986 0.85 CRHR1 (0.43) MRGPRX4RHOCRHOACCR2
SCHEMBL4923555 0.85 MRGPRX4 (0.41) MRGPRX4RHOCRHOA
SCHEMBL4932213 0.84 MRGPRX4 (0.43) MRGPRX4RHOCRHOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080221210-A1 Thyroid Receptor Agonists KARO BIO AB (SE) 2008-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080221210-A1 Thyroid Receptor Agonists TSHR, TRHR, THRA MRGPRX4 119/4885RHOC 1793/4885RHOA 1336/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.