SCHEMBL4941247

SCHEMBL4941247

Bc1ccc([N+](=O)[O-])c(C=O)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
ALOX15 P16050 1/20 0.47
PRKDC P78527 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ERN1 O75460 7/20 0.44
ALDH5A1 P51649 1/20 0.41
ABAT P80404 1/20 0.41
VCAM1 P19320 1/20 0.41
BACE1 P56817 1/20 0.39
TSHR P16473 3/20 0.38
ALDH3A1 P30838 1/20 0.38
EGFR P00533 1/20 0.38
TDP1 Q9NUW8 2/20 0.37
MAPK1 P28482 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14429392 0.85 ALDH1A1 (0.47) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL16838212 0.78 ALDH5A1 (0.59) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL1800032 0.78 ERN1 (0.65) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL8577695 0.77 CYP3A4 (0.47) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL40312 0.77 MAPK1 (0.60) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL371170 0.77 TSHR (0.62) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL274241 0.77 ERN1 (0.50) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL3894725 0.77 TDP1 (0.60) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL1014901 0.77 BACE1 (0.63) CYP3A4KDM4EALDH1A1MAPTALOX15
SCHEMBL564611 0.77 ATM (0.60) CYP3A4KDM4EALDH1A1MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012051659-A1 VIRAL POLYMERASE INHIBITORS BIOTA SCIENTIFIC MANAGEMENT PTY LTD (AU) 2012-04-26 WO disclosed
EP-2364976-A1 S1P receptor modulating compounds and use thereof EPIX Pharmaceuticals, Inc. (US) 2011-09-14 EP disclosed
WO-2009135651-A1 6-PYRIDIN-3-YL-3,4-DIHYDRO-1H-QUINOLIN-2-ONE DERIVATIVES AND RELATED COMPOUNDS AS INHIBITORS OF THE HUMAN ALDOSTERONE SYNTHASE CYP11B2 UNIVERSITÄT SAARLANDES (DE) 2009-11-12 WO disclosed