SCHEMBL4941722

SCHEMBL4941722

CS(=O)(=O)OCc1ccnc(C(=O)NC2CC2)c1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 9/20 0.60
ADORA1 P30542 3/20 0.48
PARP1 P09874 1/20 0.44
KIT P10721 1/20 0.40
BRAF P15056 1/20 0.40
KDR P35968 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
ANO1 Q5XXA6 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4307516 0.83 PARP1 (0.45) SMYD3ADORA1PARP1KITKDR
SCHEMBL12257089 0.82 SMYD3 (0.66) SMYD3ADORA1PARP1KITBRAF
SCHEMBL12233638 0.81 SMYD3 (0.61) SMYD3ADORA1PARP1KITBRAF
SCHEMBL4941679 0.81 PARP1 (0.46) SMYD3ADORA1PARP1KITBRAF
SCHEMBL4937449 0.81 LOXL2 (0.46) KITBRAF
SCHEMBL10204398 0.79 ALDH1A1 (0.45) SMYD3PARP1
SCHEMBL1166333 0.79 ALDH1A1 (0.39) SMYD3PARP1
SCHEMBL244445 0.79 SMYD3 (0.67) SMYD3ADORA1PARP1KITBRAF
SCHEMBL244667 0.78 SMYD3 (0.66) SMYD3ADORA1PARP1KITBRAF
SCHEMBL4310539 0.78 CYP4F2 (0.46) SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080293696-A1 2-Aminoarylcarboxamides Useful as Cancer Chemotherapeutic Agents BAYER PHARMACEUTICALS CORPORATION (US) 2008-11-27 US disclosed
US-20080293696-A1 2-Aminoarylcarboxamides Useful as Cancer Chemotherapeutic Agents BAYER PHARMACEUTICALS CORPORATION (US) 2008-11-27 US disclosed
US-20080293696-A1 2-Aminoarylcarboxamides Useful as Cancer Chemotherapeutic Agents BAYER PHARMACEUTICALS CORPORATION (US) 2008-11-27 US disclosed
EP-1765811-A2 2-AMINOARYLCARBOXAMIDES USEFUL AS CANCER CHEMOTHERAPEUTIC AGENTS Bayer Pharmaceuticals Corporation (US) 2007-03-28 EP disclosed
WO-2006023707-A2 2-AMINOTHIOPHENECARBOXAMIDES USEFUL AS CANCER CHEMOTHERAPEUTIC AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2006-03-02 WO disclosed
WO-2006002383-A2 2-AMINOARYLCARBOXAMIDES USEFUL AS CANCER CHEMOTHERAPEUTIC AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2006-01-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080293696-A1 2-Aminoarylcarboxamides Useful as Cancer Chemotherapeutic Agents ABCC3, HCCS, ABCC2 SMYD3 379/4885ADORA1 101/4885PARP1 834/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.