SCHEMBL4944374

SCHEMBL4944374

Cc1cc(S(C)(=O)=O)c2ncc(C(N)=O)c(Nc3cccc(Cl)c3F)c2c1

nearest known ligand 0.67

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 7/20 0.67
CSF1R P07333 11/20 0.58
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TYK2 P29597 1/20 0.42
JAK3 P52333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4948854 0.91 CSF1R (0.56) PDE4BCSF1RJAK2JAK1TYK2
SCHEMBL1275339 0.85 PDE4B (0.75) PDE4BCSF1R
SCHEMBL4949063 0.82 CSF1R (0.56) PDE4BCSF1R
SCHEMBL4951564 0.79 CSF1R (0.53) PDE4BCSF1R
SCHEMBL4949101 0.79 PDE4B (0.68) PDE4BCSF1R
SCHEMBL4952737 0.77 PDE4B (0.61) PDE4BCSF1R
SCHEMBL4949242 0.77 PDE4B (0.48) PDE4BCSF1R
SCHEMBL4951405 0.77 PDE4B (0.63) PDE4BCSF1R
SCHEMBL4952739 0.77 PDE4B (0.48) PDE4BCSF1R
SCHEMBL27649778 0.76 CSF1R (0.57) PDE4BCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633748-B1 QUINOLINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS GLAXO GROUP LTD (GB) 2008-03-05 EP claimed